Retosiban|CAS 820957-38-8|DC Chemicals

Cas No.:	820957-38-8
Chemical Name:	Retosiban
SMILES:	O=C([C@@H](C1CC2=C(C=CC=C2)C1)N3)N([C@H](C4=COC(C)=N4)C(N5CCOCC5)=O)[C@H]([C@H](CC)C)C3=O
Formula:	C₂₇H₃₄N₄O₅
M.Wt:	494.58
Sotrage:	Please store the product under the recommended conditions in the Certificate of Analysis.

Cat. No.	Product name	Field of application
DC47258	Carbetocin acetate	Carbetocin acetate, an oxytocin (OT) analogue, is an oxytocin receptor agonist with a Ki of 7.1 nM. Carbetocin acetate has high affinity to chimeric N-terminus (E1) of the oxytocin receptor (Ki=1.17 μM). Carbetocin acetate has the potential for postpartum hemorrhage research. Carbetocin acetate can crosse the blood-brain barrier and produces antidepressant-like activity via activation of oxytocin receptors in the CNS.
DC46970	L-372662	L-372662 is a potent and orally active non-peptide oxytocin antagonist with a Ki value of 4.8. The Kd value of L-372662 for wild-type hOTR and [A318G]OTR is 5.8 nM and 73 nM. L-372662 shows selectivity to OTR:V1aR.
DC45573	[Asp5]-Oxytocin	[Asp5]-Oxytocin is the first 5-position neurohypophyseal hormone analogue possessing significant biological activity.
DC41072	Retosiban	Retosiban (GSK221149A) is a potent and selective oxytocin antagonist with a Ki of 0.65 nM.