YY-20394|PI3K inhibitor

Cas No.:	1702816-75-8
Chemical Name:	Linperlisib
Synonyms:	PI3Kδ-IN-2;pi3Kdelta-IN-2;PI3K(delta)-IN-2;Linperlisib HCl;Linperlisib free base;05HYK3CV9N;PI3K;A-IN-2;Methanesulfonamide, N-(5-(6-fluoro-8-((4-(1-hydroxy-1-methylethyl)-1-piperidinyl)methyl)-2-(4-morpholinyl)-4-quinazolinyl)-2-methoxy-3-pyridinyl)-;N-[5-[6-fluoro-8-[[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl]-2-morpholin-4-ylquinazolin-4-yl]-2-methoxypyridin-3-yl]methanesulfonamide;N-{5-[6-fluoro-8-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl;Linperlisib;YY-20394
SMILES:	S(C([H])([H])[H])(N([H])C1=C(N=C([H])C(=C1[H])C1C2=C([H])C(=C([H])C(=C2N=C(N=1)N1C([H])([H])C([H])([H])OC([H])([H])C1([H])[H])C([H])([H])N1C([H])([H])C([H])([H])C([H])(C(C([H])([H])[H])(C([H])([H])[H])O[H])C([H])([H])C1([H])[H])F)OC([H])([H])[H])(=O)=O
Formula:	C₂₈H₃₇FN₆O₅S
M.Wt:	588.6940
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	YY-20394(PI3Kδ-IN-2) is a potent and selective inhibitor of PI3Kδ extracted from patent WO 2015055071 A1, compound 10; has an IC50 of 6.4 nM.
Target:	PI3Kδ:6.4 nM (IC50)
References:	[1]. WO 2015055071 A1

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YY-20394(PI3Kδ-IN-2)