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GSK256073

Cat. No.: DC42499

Chemical Structure

862892-90-8

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Field of application

GSK256073 is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM)and dyslipidemia. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2

Chemicals Properties Biological activity Related products COA MSDS Datasheet

Cas No.:	862892-90-8
Synonyms:	GSK256073
SMILES:	O=C(N(C1=C2NC(Cl)=N1)CCCCC)NC2=O
Formula:	C₁₀H₁₃ClN₄O₂
M.Wt:	256.69
Sotrage:	Powder -20°C 3 years 4°C 2 years In solvent -80°C 6 months -20°C 1 month

Cat. No.	Product name	Field of application
DC42499	GSK256073	GSK256073 is a potent, selective and orally active GPR109A agonist and a long-lasting and non-flushing HCA2 full agonist with a pEC50 of 7.5 (human HCA2). GSK256073 acutely improves glucose homeostasis via inhibition of lipolysis and has the potential for the study of type 2 diabetes mellitus (T2DM)and dyslipidemia. GPR109A: G-protein coupled receptor 109A; HCA2: hydroxy-carboxylic acid receptor 2
DC9455	MK-6892	MK-6892 is a highly potential GPR109A agonist with Ki value of 4.0 nM.

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