Demethoxyviridiol is a mycotoxin that inhibits phosphatidylinositol 3-kinase (PI3K).

Tenellin is a fungal metabolite that inhibits Mg2±, Ca2±, and Na+/K±ATPase activities in erythrocytes. Tenellin is cytotoxic to Sf9 and Sf21 insect cells.

Steffimycin B is an anthracycline bacterial metabolite. It binds to DNA, preferentially intercalating at sites containing cytosine and guanine. Steffimycin B is cytotoxic to MCF-7, KB, NCI-H187, and Vero cells. It is active against M. tuberculosis, B. cereus, and P. falciparum.

Imidocarb propionate is an antiprotozoal agent that eliminates blood parasites. Formulations containing imidocarb have been used in the veterinary treatment of babesiosis and other protozoal infections.

GHV sodium salt is a sedative and active metabolite of γ-valerolactone.

(-)-Bicuculline methochloride is an enantiomer of the GABA antagonist (+)-bicuculline methochloride. It increases the firing rate in rat cortical neurons similar to the (+) isomer but lacks GABA antagonist activity. (-)-Bicuculline methochloride inhibits sodium-independent GABA receptor binding with an IC50 value of 500 μM, which is approximately 100-fold less potent than (+)-bicuculline methochloride, but there is no stereoselectivity for sodium-dependent GABA receptor binding.

4β-Hydroxywithanolide E is a withanolide steroidal lactone that has anti-inflammatory and anticancer activities. It inhibits LPS-induced nitric oxide (NO) production and TNF-α-induced NF-κB activity. 4β-Hydroxywithanolide E inhibits LPS-induced increases in inducible nitric oxide synthase (iNOS) and COX-2 levels and Akt and STAT1 phosphorylation. It inhibits Wnt signaling in HCT116 and SW480 colorectal cancer cells (IC50s = 1.85 and 2.67 μM, respectively).3 4β-Hydroxywithanolide E inhibits the proliferation of HCT116, SW480, HT-29, and LoVo cells.

Oxychlororaphine is a phenazine microbial metabolite that has been found in a variety of bacteria and has anticancer, antibacterial, and antifungal activities. It is cytotoxic to A549, HeLa, and SW480 cancer cells. Oxychlororaphine halts the cell cycle at the G1 phase and induces apoptosis in A549 cells. It is active against Streptomyces bacteria and T. mentagrophytes, E. floccosum, C. albicans, M. audouini, and B. dermatitidis fungi.

(R)-Aminoglutethimide tartrate is an anticancer drug that belongs to the family of drugs called nonsteroidal aromatase inhibitors. Aminoglutethimide is used to decrease the production of sex hormones (estrogen in women or testosterone in men) and suppress the growth of tumors that need sex hormones to grow.

(S)-Aminoglutethimide is an anticancer drug that belongs to the family of drugs called nonsteroidal aromatase inhibitors. Aminoglutethimide is used to decrease the production of sex hormones (estrogen in women or testosterone in men) and suppress the growth of tumors that need sex hormones to grow.

(D)-Aminoglutethimide is a nonsteroidal aromatase inhibitors. Aminoglutethimide is used to decrease the production of sex hormones (estrogen in women or testosterone in men) and suppress the growth of tumors that need sex hormones to grow.

Fluprostenol, (+)-, is an analog of Prostaglandin F2α with potent FP receptor agonist activity.

Benzylurea is a competitive inhibitor of cytokinin oxidase/dehydrogenase.

Ethylenediaminediacetic acid (EDDA) is a derivative of two molecules of glycine wherein the amines are linked.

Aureothricin is a dithiolopyrrolone antibiotic that exhibits broad-spectrum antimicrobial activity against many Gram-positive and Gram-negative bacteria as well as strains of M. tuberculosis. It is also reported to inhibit tumor angiogenesis, blocking activity of the vitronectin receptor integrin αvβ3.

Metoprolol acid is a pharmacologically inactive urinary metoprolol metabolite.

Agroclavine is a clavine type of ergot alkaloid with D1 dopamine and a-adrenoceptor agonistic properties.

Triprolidine hydrochloride anhydrous is a Histamine H1 antagonist used in allergic rhinitis, asthma, and urticaria.

Averantin is an Aflatoxin B(1) precursor.

Avarone is a cytostatic agent which has potent antileukemic activity in vitro. Avarone also displays antibacterial and antifungal activities against a limited range of microorganisms.

Avarol induces apoptosis in pancreatic ductal adenocarcinoma cells by activating PERK-eIF2α-CHOP signaling. Avarl also acts as a competitive AChE inhibitor which are non-hepatotoxic and neuroprotective agents for Alzheimer's disease.

Chlortetracycline is a broad-spectrum antibiotic tetracycline with a 7-chloro substitution. It inhibits growth of both Gram-positive and Gram-negative bacteria. It acts by inhibiting protein synthesis.

Aseanostatin P5 inhibits myeloperoxidase (MPO) release from human polymorphonuclear leukocytes.

Heptaminol hydrochloride is an amino alcohol used as a myocardial stimulant, vasodilator, and to relieve bronchospasm. Its most common therapeutic use is in orthostatic hypotension. The mechanism of heptaminol's therapeutic actions is not well understood although it has been suggested to affect catecholamine release or calcium metabolism.

(±)-Shikonin is a naphthazarin with antineoplastic and angiogenesis inhibiting activities.

Ibuprofen lysine is a non-steroidal anti-inflammatory drug (NSAID). The lysine suspension of Ibuprofen may act more quickly and effectively than base Ibuprofen.

Arbaprostil is a synthetic prostaglandin E analog that protects gastric mucosa, prevents ulceration, and promotes healing of peptic ulcers. The protective effect is independent of acid inhibition. It is also a potent inhibitor of pancreatic function and can inhibit the growth of experimental tumors. Arbaprostil is a prodrug for the potent PGE2.

Apomorphine hydrochloride is a Dopamine (D1 and D2) receptor agonist which may be effective in the treatment of Parkinson's disease.

Methylthiouracil is thiourea antithyroid agent that inhibits the synthesis of thyroid hormone. It is used in the treatment of hyperthyroidism.

Amisometradine is a diuretic which may be used in the treatment of congestive heart failure.