Potent PARP inhibitor

Novel selective non-steroidal agonist of G-protein bile acid receptor 1 (GPBAR1, also known as TGR5 or M-BAR)

Curcumin analog, exhibiting potent growth suppressive activity in human colorectal carcinoma cells

Natural potent inducer of apoptosis in MCF-7 cell lines

Antipsychotic and cognitive enhancer; Dopamine D1 and D2 receptor modulator

Natural inhibitor of Musashi family of RNA-binding proteins

Agonist of the GnRH receptor, inducing the secretion of the gonadotropins follicle-stimulating hormone and luteinizing hormone from the pituitary gland and to increase sex hormone production by the gonads

Dual Glycolate Oxidase/Lactate Dehydrogenase A (GO/LDHA) Inhibitor for Primary Hyperoxaluria

Novel potent GNMT inducer, inhibiting Huh7 cell growth in vitro and xenograft in vivo

Novel inhibitor of Gram-negative lipoprotein trafficking

Natural highly potent HIV latency-reversing agent

Dose dependent up-regulator of the level of E-cadherin in SW620 cells

Novel inhibitor of Plasmodium falciparum, killing both blood- and sexual-stage P. falciparum parasites

Novel Inhibitor of EGF-EGFR Interactions

Novel potent aryl hydrocarbon receptor (AHR) antagonist with the capacity to inhibit both DRE-dependent and -independent activity

Novel selective CHK1 inhibitor

Novel GluN2A-selective NMDA receptor positive allosteric modulator (PAM)

Negative control for GNE-2256

Novel inhibitor of nicotinamide phosphoribosyl transferase (NAMPT)

Novel NMDAR PAM with both an improved pharmacokinetic profile and increased selectivity against AMPARs

Novel GluN2A-selective NMDA receptor positive allosteric modulator (PAM)

Novel Met inhibitor

Novel potent and selective RORc inverse agonist

Novel GluN2A subunit-selective and brain-penetrant positive allosteric modulator (PAM) of The N-methyl-d-aspartate receptor (NMDAR)

Novel Tubulin Polymerization Inhibitor

Negative control for GMB-805

Novel potent BCR-Abl PROTAC, inducing degradation and demonstrating in vivo activity

Selective modulator of gamma-aminobutyric acid(A) receptors

Novel GM3 derivative, showing excellent migration and invasion inhibitory effects in cells and marked antitumor activity in C57BL/6 mice, involving focal adhesion and ECM-receptor interaction signaling pathways

Metabolite of soy isoflavones, promoting the proliferation of bone marrow stromal cells and osteoblasts and suppresses bone turnover