Novel ligand of voltage-gated calcium channel α2δ-1 subunit (Cavα2δ-1)

Novel selective reversible inhibitor of cathepsin X

Selective inhibitor of cathepsin B endopeptidase and exopeptidase activities

Selective inhibitor of cathepsin B endopeptidase and exopeptidase activities

Novel activator of autophagy for potential treatment of cystic fibrosis

Natural potent neutrophil elastase (NE) inhibitor with an IC 50 value of 2.79 ± 0.07 μM

The first inhibitor of fungal (1→3)-β-D-glucan synthesis

Novel Cas9 Inhibitor, direct binding to apo-Cas9, preventing Cas9:gRNA complex formation

DNA minor groove alkylating agent, alkylating N3 of adenine in a consensus sequence 5'-(A/T)(A/T)A*

Irreversible and nonselective Monoamine_oxidase_inhibitor>monoamine oxidase inhibitor (MAOI)

Novel orally available α4 integrin receptor inhibitor

Long acting ß2-adrenoreceptor agonist (LABA)

Anthracycline antineoplastic antibiotic, intercalating into DNA and interacting with topoisomerase II, thereby inhibiting DNA replication and repair and RNA and protein synthesis.

Novel, potent, long-acting, selective, orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4) with hypoglycemic activity

Novel potent inhibitor of coactivator-associated arginine methyltransferase 1 (CARM1)

Novel inhibitor of full-length GST-tagged CARM-1

Inducer of deformation in Zebrafish>Zebrafish through the AhR-mediated, CYP1A-independent pathway

Novel fluorescent probe targeting of G-quadruplex structures and trapping cytoplasmic RNA G-quadruplex structures in cells

Mixture of Meropenem and vaborbactam for adults with complicated urinary tract infections (cUTI), including a type of kidney infection, pyelonephritis, caused by specific bacteria

Antioxidant, free radical scavenger and potent inhibitor of lipid peroxidation

Antimuscarinic and anticholinergic, acting as an antagonist of NMDA receptor

Broad spectrum antibiotic used in the therapy of drug resistant tuberculosis as a second line agent

Reverse-transcriptase_inhibitor>Non-nucleoside reverse transcriptase inhibitor

Novel self-assembling lysine-rich cationic amphipathic peptide (CAP)

Natural cannabinoid precursor

Natural cannabinoid precursor

Novel destabilizer of CAND1-Cullin1 interaction, inducing a p53-stress response pathway

Transmembrane protease serine 2 (TMPRSS2) inhibitor for the treatment of chronic pancreatitis and postoperative gastric reflux, blocking SARS-CoV-2 replication in TMPRSS2-expressing human cells

Ionophore highly selective for Ca , potentiating responses to NMDA but not quisqualate

Dual inhibitor of fibroblast growth factors (FGF) and vascular endothelial growth factor (VEGF) ; Anti-angiogenic