Pargyline is an irreversible selective monoamine oxidase (MAO)-B inhibitor drugwith antihypertensive properties. Pargyline has been found to bind with high affinity to the I2 imidazoline receptor (an allosteric site on the MAO enzyme).

Chlorphenoxamine HCl is an antihistaminic agent which reverses multidrug resistance in L1210 tumor cells.

Gentamicin X2 Sulfate is a potent premature stop codon readthrough molecule and the common precursor of the gentamicin C antibiotic complex.

Vicriviroc Malate is a potent, highly selective, and orally bioavailable CCR5 antagonist.

Norfluoxetine hydrochloride is an active metabolite of fluoxetine.

MP265 is an inhibitor of MreB polymerization.

Cellocidin is a potent growth inhibitor for gammaherpesvirus-associated B-lymphomas that acts through activation of both the NF-κB and c-Myc-mediated signaling pathways.

GSNO is an endogenous transnitrosation donor involved in S-nitrosation of a variety of cellular proteins. It acts by regulating diverse protein functions

NP-313 is an antithrombotic agent with dual inhibition of thromboxane A2 synthesis and calcium entry.

5-Methylcytosine is a methylated cytosine. It acts as a ligand of the hDNMT1.

Cytidine 5'-diphosphate disodium is a substrate of CDP (nucleoside diphosphate) kinase (2.7.4.6). It has been shown to produce CTP in support of DNA and RNA biosynthesis and of ribonucleotide reductase to produce dCMP.

Sodium Oxamate is an LDH inhibitor. It inhibits L(+)-lactate dehydrogenase and derails the entire gluconeogenic pathway.

Propentofylline is a phosphodiesterase inhibitor with neuroprotective effect. It was studied for the treatment of Alzheimer's disease and multi-infarct dementia, as well as its action as an adenosine reuptake inhibitor.

Piretanide is a time- and voltage-dependent blocker of CFTR Cl(-) currents. It also acts as a loop diuretic.

GMQ hydrochloride is a potent and selective modulator of acid-sensing ion channel (ASIC). It activates ASIC3 channels under neutral pH and blocks acid-induced maximal peak current.

ROPA, also known as Resiniferonol 9,13,14-ortho-phenylacetate, is a potent PKCalpha and PKCgamma activator that promotes tumor growth through PKC-activation.

SXT1596 is a novel inhibitor of the SS18-SSX/TLE1 interaction. SXT1596 decreases cell viability and reactivates EGR1 expression in synovial sarcoma.

2-Arachidonoylglycerol is an endocannabinoid, an endogenous agonist of the CB1 receptor. At a concentration of 0.3nM, 2-Arachidonoylglycerol induces a rapid, transient increase in intracellular free calcium in NG108-15 neuroblastoma X glioma cells through a CB1 receptor-dependent mechanism.

Pentetrazol, also known as pentylenetetrazole, metrazol, pentetrazol (INN), pentamethylenetetrazol, Corazol, Cardiazol or PTZ, is a non-competitive GABA antagonist. It was formerly used as a drug for circulatory and respiratory stimulation.

4-POBN is a potent and irreversible inhibitor of myeloperoxidase.

U-0521 is a catechol-O-methyltransferase (COMT) inhibitor. U-0521 enhances the availability and utilization of levodopa in the brain.

Isomaltitol, also known as Palatinit or Isomalt, is a sugar alcohol. Isomaltitol is commonly used as a sweetener in food products. There is some evidence that Isomaltitol could be used to aid mucus clearance in cystic fibrosis patients.

Benzetimide HCl, also known as EINECS 227-072-8, Spasmentral, and Dioxatrine, is a muscarinic acetylcholine receptor antagonist. Benzetimide HCl has been used to treat neuroleptic-induced parkinsonism. Benzetimide is an enantiomer of dexetimide.

Senecioic acid is a crystalline unsaturated fatty acid found in the pheromones of mealybug species.

Heptelidic acid is an esquiterpene lactone produced by the fungus T. koningii with antibiotic activity against anaerobic bacteria such as Bacteroides. It acts as an irreversible inhibitor of GAPDH that binds to the cysteine-149 residue at the active site of the enzyme.

Chromotrope 2B is a reagent for boric acid and borates.

3-Benzoylpyridine is a decomposition product of the soman antidote HGG-12.

Exifone is a bioactive chemical.

Boldine is an alkaloid of the aporphine class that can be found in the boldo tree and in Lindera aggregata. Boldine has antioxidant activity that effectively protects against free radical induced lipid peroxidation or enzyme inactivation. In addition, it has alpha-adrenergic antagonist activities in vascular tissue, and it has also been reported to have hepatoprotective, cytoprotective, antipyretic and anti-inflammatory effects.

Norethindrone acetate is used in combination with estrogen as a contraceptive (oral). It is reasonably anticipated to be a human carcinogen.