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GR-127935 hydrochloride

  Cat. No.:  DC21064   Featured
Chemical Structure
148642-42-6
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More than 5000 active chemicals with high quality for research!
Field of application
GR-127935 potent and selective 5-HT1B/1D receptor antagonist with pKi of 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptor.
Chemicals PropertiesBiological activity Related products COA MSDS Datasheet
Cas No.: 148642-42-6
Chemical Name: N-[4-methoxy-3-(4-methylpiperazin-1-yl)phenyl]-4-[2-methyl-4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]benzamide hydrochloride
Synonyms: GR127935
SMILES: Cl.CN1CCN(C2C=C(NC(C3C=CC(C4C=CC(C5=NOC(C)=N5)=CC=4C)=CC=3)=O)C=CC=2OC)CC1
Formula: C29H31N5O3.HCl
M.Wt: 534.06
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: GR-127935 potent and selective 5-HT1B/1D receptor antagonist with pKi of 8.5 for both guinea pig 5-HT1D and rat 5-HT1B receptor.
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