Novel Potent Dual AChE/GSK-3 Inhibitor for the Treatment of Alzheimers Disease

Novel Irriversible Inhibitor of Parasite Motility and Invasion

Novel Inhibitor of Parasite Motility and Invasion

Novel Inhibitor of Parasite Motility and Invasion

Natural radical scavenger on ABTS

Novel inhibitor of the catalytic functions of peroxiredoxin (Prx) and thioredoxin (Trx) systems

Inhibitor of HIV-1 Assembly that Targets the Phosphatidylinositol (4,5)-bisphosphate Binding Site of the HIV-1 Matrix Protein

Novel Inhibitor of Adenovirus Gene Transfer

Novel Inhibitor of Adenovirus Gene Transfer

Novel inhibitor of the type III secretion system (T3SS), acting as a anti-microbial agent against Xanthomonas oryzae pv. oryzae (Xoo)

Type-A trichothecene mycotoxin

Selective class D inhibitor of the Ca -activated Cl- Channel, Ano1(TMEM16A)

Selective class B inhibitor of the Ca -activated Cl- Channel, Ano1(TMEM16A)

Novel potent PPARγ antagonist with much improved drug-like properties and promising pharmacokinetic profile

Potent and selective CCKA receptor antagonist

Novel COX-2 inhibitor

Potent inhibitor of both rodent and human MAO-B, proved to be safe in high doses with no hERG and mutagenic activities and demonstrated neuroprotection in an in vivo chronic model of PD

K+ channel blocker

Novel microtubule-stablizer

Novel Mycobacterium tuberculosis growth inhibitor

Negative control of Syn-1 peptide, having the same amino acid composition as Syn-1 peptide, but a scrambled sequence

Novel potent and specific inhibitor of syncytin-mediated cell fusion, completely blocking cell fusion at 1.6 μg/ml

Novel inhibitor of the Syk kinase (spleen tyrosine kinase)

Novel universal opioid receptor agonist

Novel highly potent and selective CDK7 inhibitor, demonstrating broad anti-tumor activity in vivo

Novel selective OXE receptor antagonist

Potent differentiating agent

Natural potent alpha-mannosidase inhibitor, exhibiting antimetastatic, antiproliferative, and immunomodulatory activities

Novel clickable tumor-specific irreversible inhibitor of stearoyl CoA desaturase (SCD)

D2 dopamine receptor partial agonist in adenylyl cyclase inhibition assay and antagonist in the GIRK and phospho ERK1/2 assays