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| Cat. No. | Product Name | Field of Application | Chemical Structure |
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| DC33597 | BIBF0775 Featured |
BIBF0775 is an inhibitor of the transforming growth factor β receptor I (TGFβRI). X-ray structure analysis showed that BIBF0775 soaked into the kinase domain of TGFβRI.
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| DC33602 | QBS(CU242) Featured |
QBS(CU-242) or 2-Amino-N-quinolin-8-yl-benzenesulfonamide, is an Inhibitor of cell cycle at G2 phase; apoptosis inducer. NUN82647 has CAS#16082-64-7, and inchi key: NIOOKXAMJQVDGB-UHFFFAOYSA-N. According to Hodoodo Chemical Nomenclature, It is named: NUN-82647.
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| DC22582 | AS601245 Featured |
AS601245 is an orally active, selective, ATP competitive JNK (c-Jun NH2-terminal protein kinase) inhibitor with IC50s of 150, 220, and 70 nM for three JNK human isoforms (hJNK1, hJNK2, and hJNK3), respectively. AS601245 exhibits 10- to 20-fold selectivity over c-src, CDK2, and c-Raf and more than 50- to 100-fold selectivity over a range of Ser/Thr- and Tyr-protein kinases. Neuroprotective properties.
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| DC12129 | 1F-Fructofuranosylnystose Featured |
1F-Fructofuranosylnystose can be used in the synthesis of Fructooligosaccharides (FOSs). Fructooligosaccharides exhibit lots of beneficial effects on our health and have been used as food ingredients.
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| DC21521 | PNU-112455A Featured |
PNU-112455A is an ATP-competitive CDK2/5 inhibitor with Ki of 2 uM and 2 uM for cdk2·GST-cyclin E and cdk5·GST-p25 respectively, shows no activity against c-c-Met, IGR-1R, and ERK2..
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| DC9220 | 1-Kestose Featured |
1-Kestose is a fructo-oligosaccharide (FOS) with prebiotic properties, and is a polymer of d-fructose joined by β(2→1) linkages and terminated with a d-glucose molecule linked to fructose by an α(1→2) bond as in sucrose.
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| DC10889 | 1-NA-PP 1 hydrochloride Featured |
1-Naphthyl PP1(1-NA-PP1) is a selective inhibitor of src family kinases v-Src and c-Fyn as well as the tyrosine kinase c-Abl.
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| DCAPI1534 | Alfacalcidol Featured |
1α-Hydroxyvitamin D3 is a form of vitamin D that helps the body absorb calcium from food.
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| DC9647 | 20-Deoxyingenol Featured |
20-Deoxyingenol is a natural compound.
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| DC8419 | SB-334867 Featured |
SB-334867 is a selective orexin-1 (OX1) receptor antagonist.
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| DC33300 | L-765314 Featured |
L-765,314 is a drug which acts as a potent and selective antagonist for the Alpha-1 adrenergic receptor subtype α1B. It has mainly been used to investigate the role of α1B receptors in the regulation of blood pressure.
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| DC9802 | 23-hydroxy butulinic acid (23-HBA) Featured |
23-hydroxy butulinic acid (23-HBA) is a potent angiogenesis inhibitor.
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| DC22871 | MS-402 Featured |
MS402 is a BD1-selective BET BrD inhibitor with Kis of 77 nM, 718 nM, 110 nM, 200 nM, 83 nM, and 240 nM for BRD4(BD1), BRD4(BD2), BRD3(BD1), BRD3(BD2), BRD2(BD1) and BRD2(BD2), respectively. MS402 blocks Th17 cell differentiation and ameliorates colitis in mice.
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| DC32382 | Brassinazole Featured |
Brassinazole is an inhibitor of brassinosteroid biosynthesis that has been developed in order to probe the myriad functions of brassinosteroids.
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| DC31005 | GRP-60367 Featured |
GRP-60367 is a first-in-class direct-acting RABV inhibitor with EC50 from 2 to 52 nM (different host cell lines) that blocks RABV G protein-mediated viral entry.
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| DC20155 | Tegoprazan Featured |
Tegoprazan, a potassium-competitive acid blocker, is a potent, oral active and highly selective inhibitor of gastric H+/K+-ATPase that could control gastric acid secretion and motility, with IC50 values ranging from 0.29-0.52 μM for porcine, canine, and human H+/K+-ATPases in vitro.
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| DC23041 | Isochlorogenic acid A Featured |
3,5-Dicaffeoylquinic acid (3,5-DCQA) is a natural phenolic compound that has been found in L. japonica, I. kaushue, and other plants.It has antioxidant, anti-inflammatory, and antiviral biological activities.
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| DC10404 | BIA 10-2474 Featured |
BIA 10-2474 is an inhibitor of fatty acid amide hydrolase (FAAH) with IC50 values of 50 to 70mg/kg in various rat brain regions.
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| DC28671 | DT2216 Featured |
DT2216 is a selective B-cell lymphoma extra large (BCL-XL) proteolysis-targeting chimera (PROTAC). DT2216 targets BCL-XL to the Von Hippel-Lindau (VHL) E3 ligase for degradation. DT2216 inhibits various BCL-XL-dependent leukemia and cancer cells but considerably less toxic to platelets.
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| DC10861 | 3BDO Featured |
3BDO is a new mTOR activator which can also inhibit autophagy.
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| DC39825 | JC-1 Featured |
JC-1 is a membrane-permeable cationic dye that is used to study mitochondrial integrity in the context of cellular apoptosis.
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| DC12491 | 3-methyl toxoflavin Featured |
3-methyl toxoflavin. Toxoflavin acts as a pH indicator, changing between yellow and colorless at pH 10.5.
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| DC12664 | 3-pyridine toxoflavin Featured |
3-pyridine toxoflavin is an impurity of toxoflavin.
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| DC8245 | 4E1rcat Featured |
4E1RCat is an inhibitor of protein translation that has been shown to prevent eIF4E:eIF4G and eIF4E:4E-BP1 interaction.
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| DC10689 | 4P-PDOT Featured |
4P-PDOT, also known as 4-phenyl-2- propionamidotetralin, is a MT2-receptor-specific antagonist. MT2 melatonin receptor may be a novel target for analgesic drug development.
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| DC7592 | 4SC-202 Featured |
4SC-202 is an orally bioavailable benzamide and inhibitor of human class I histone deacetylases (HDACs) isoenzymes 1, 2 and 3, with potential antineoplastic activity. HDAC inhibitor 4SC-202 selectively binds to and inhibits class I HDACs leading to an acc
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| DC10877 | 5,3-AB-CHMFUPPYCA Featured |
5,3-AB-CHMFUPPYCA is an analytical reference standard that is structurally classified as a synthetic cannabinoid.
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| DC9371 | 5-FAM SE Featured |
5-FAM SE is a single isomer, it is one of the most popular green fluorescent reagents used for labeling peptides, proteins and nucleotides.
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| DC9372 | 6-FAM SE Featured |
6-FAM SE is another isomer of carboxyfluorescein.
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| DC10854 | 6-MITC Featured |
6-MITC is an inhibitor of viability of both PANC-1 and BxPC-3 cells. It also acts as an inhibitor of the expression of CSC signaling molecule SOX2.
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