Activator of SHIP-1

Cyclooxygenase Inhibitor and Prostagladin Synthase Inhibitor

Novel caged glutamate

Antineoplastic agent, alkylating and crosslinking DNA, resulting in DNA strand breaks and inhibition of DNA and RNA synthesis

Mycotoxin with antibiotic and carcinogenic activity

Antibiotic, a natural penicillin, synthesized in vitro by incubating (S-octanoyl)glutathione, 6-APA and AT

Novel potent and broad-spectrum anti-influenza A virus (anti-IAV) activities with low risk of inducing drug resistance

Inhibitor of calcium-dependent complex formation with p53 [(Ca)S100B-p53] in malignant melanoma (MM), restoring p53 tumor suppressor activity in vivo

Innate defense regulator, target stringent response-controlled virulence in a Pseudomonas aeruginosa murine cutaneous infection model

ApoA-I/HDL mimetic peptide, efficiently crossing the blood-brain barrier and modulating amyloid beta distribution between brain and plasma

Broad-spectrum virus- and host-targeting peptide, inhibiting coronaviruses and other respiratory viruses

Agonist of dopamine receptor subtypes D1 and D2

Exceptionally Potent and Membrane-Embedded Inhibitor of Bilayer Lipid Peroxidation

Non-sulfhydryl angiotensin converting enzyme (ACE) inhibitor

Novel allosteric inhibitor of E. coli Hsp70 (DnaK) and human Hsp70 proteins

First Inhibitor of PEX14-PEX5 Protein-Protein Interaction (PPI) with Trypanocidal Activity

Novel γ-secretase inhibitor

Dose dependent inhibitor of multiple fibrotic genes

Selective dopamine D3/D2 receptor antagonist

Novel potent and selective PDE8B/8A inhibitor

Irriversible inhibitor of kynurenine amino transferase II (KAT II)

Novel selective hTRPV4 Antagonist (hTRPV4 IC50 49nM; rTRPV4 IC50 1,150nM)