| Cat. No. | Product Name | Field of Application | Chemical Structure |
|---|---|---|---|
| DC11364 | Levocetirizine；(R)-Cetirizine (hydrochloride) | (R)-Cetirizine is the (R)-enantiomer of the histamine H1 receptor antagonist and second generation antihistamine cetirizine. |
|
| DC10279 | Acrivastine | Acrivastine (BW825C) is a short acting histamine 1 receptor antagonist for the treatment of allergic rhinitis. |
|
| DCAPI1467 | Alcaftadine | Alcaftadine |
|
| DC9469 | Azatadine (dimaleate) | Azatadine dimaleate is an histamine and cholinergic inhibitor with IC50 of 6.5 nM and 10 nM, respectively. |
|
| DC9130 | Azelastine HCl | Azelastine HCl is a potent, second-generation, selective, histamine antagonist. |
|
| DCAPI1500 | Bepotastine Besilate Featured | Bepotastine Beslilate (Bepreve) is a histamine H1 receptor anatagonist. |
|
| DC8898 | Bepotastine Featured | Bepotastine is a non-sedating, selective antagonist of the histamine 1 (H1) receptor. |
|
| DC8967 | Betahistine Dihydrochloride | Betahistine Dihydrochloride is a histamine H3 receptors inhibitor used as an antivertigo drug. |
|
| DC8830 | Betahistine Featured | Betahistine is a strong affinity histamine H3 receptor antagonist and weak affinity agonist of histamine H1 receptors. |
|
| DC7995 | Bilastine Featured | Bilastine is a selective histamine H1 receptor antagonist used for treatment of allergic rhinoconjunctivitis and urticaria. |
|
| DC9141 | Brompheniramine hydrogen maleate | Brompheniramine maleate is a histamine H1 receptors antagonist. |
|
| DC10222 | CarbinoxaMine Maleate | Carbinoxamine maleate is a histamine-H1 receptor blocking agent with antihistamine and anticholinergic properties. |
|
| DC9154 | Cetirizine 2HCl | Cetirizine 2Hcl, a second-generation antihistamine, is a major metabolite of hydroxyzine, and a racemic selective H1 receptor inverse agonist used in the treatment of allergies, hay fever, angioedema, and urticaria. |
|
| DC9111 | Chlorpheniramine Maleate | Chlorpheniramine maleate is an histamine H1 receptor antagonist with IC50 of 12 nM. |
|
| DC9062 | Chlorprothixene | Chlorprothixene has strong binding affinities to dopamine and histamine receptors, such as D1, D2, D3, D5, H1, 5-HT2, 5-HT6 and 5-HT7, with Ki of 18 nM, 2.96 nM, 4.56 nM, 9 nM, 3.75 nM, 9.4 nM, 3 nM and 5.6 nM, respectively. |
|
| DC9002 | Cimetidine | Cimetidine is a histamine-2 (H2) receptor antagonist. |
|
| DC9896 | Cinnarizine Featured | Cinnarizine is a medication derivative of piperazine, and characterized as an antihistamine and a calcium channel blocker. |
|
| DC2062 | Ciproxifan (FUB-359) Featured | Ciproxifan is an antagonists of H3-type histamine receptors. |
|
| DC9466 | Ciproxifan (maleate) Featured | Ciproxifan maleate(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity at other receptor subtypes. |
|
| DC11048 | Contilisant | Contilisant is a neuroprotective, non-toxic, antioxidant, permeable ligand, showing in vitro pharmacological properties on the selected biological targets (hAChE IC50=0.53 uM. |
|
| DCAPI1536 | Cyproheptadine Hydrochloride | Cyproheptadine hydrochloride is a migraine prophylactic and Non-selective SR-2A (5HT2) antagonist. Cyproheptadine hydrochloride is an inhibitor of Histamine H1 Receptor and SR-2C. |
|
| DC9057 | Desloratadine | Desloratadine(Sch34117) is a potent antagonist for human histamine H1 receptor used to treat allergies. |
|
| DC4161 | Dimebon dihydrochloride | Dimebon is an antihistamine drug. |
|
| DC9109 | Doxylamine succinate | Doxylamine is a first generation antihistamine; can be used by itself as a short-term sedative and in combination with other drugs to provide night-time allergy and cold relief. |
|
| DC9467 | Epinastine Featured | Epinastine(WAL801) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis. |
|
| DC9073 | Famotidine | Famotidine is a competitive histamine H2-receptor antagonist. Its main pharmacodynamic effect is the inhibition of gastric secretion. |
|
| DC9175 | Fexofenadine Hydrochloride Featured | Fexofenadine is a third-generation antihistamine pharmaceutical drug used in the treatment of allergy symptoms, such as hay fever, nasal congestion, and urticaria. |
|
| DC10102 | GSK189254A Featured | GSK189254A (GSK189254) is a novel, potent and selective histamine H3 receptor antagonist with pKi values of 9.59-9.90 and 8.51-9.17 for human and rat H3, respectively. |
|
| DC12266 | H4 Receptor antagonist 1 | H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM. |
|
| DC11328 | Hydroxyzine | Hydroxyzine is a histamine H1 receptor antagonist (Ki = 1.9 nM). |
|
