GABA Receptor

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Cat. No.	Product Name	Field of Application
DC10625	(+)-Bicuculline Featured	(+)-Bicuculline is a competitive antagonist of GABAA receptors with IC50 of 2 μM, also blocks Ca(2+)-activated potassium channels.
DC9450	(R)-Baclofen	(R)-Baclofen(STX209) is a selective GABAB receptor agonist.
DC9026	Afloqualone	Afloqualone is a agonist of GABA receptor .
DC9764	Afoxolaner Featured	Afoxolaner is an isoxazoline that inhibits insect and acarine ligand-gated chloride channels, in particular those gated by the neurotransmitter gamma-aminobutyric acid (GABA), blocking pre and post synaptic transfer of chloride ions across cell membranes.
DC10311	Allopregnanolone Featured	Allopregnanolone is a progesterone metabolite. Allopregnanolone is an allosteric modulator of the GABA receptor.
DC11657	PPT(Propyl pyrazole triol ) Featured	Propyl pyrazole triol (PPT) is a selective estrogen receptor alpha (ERα) agonist. The relative binding affinity of Propyl pyrazole triol for ERα (ERα: 49%) around 410 times higher compared with estrogen receptor beta (ERβ: 0.12%).
DC8971	Baclofen	Baclofen is a gamma-amino-butyric acid (GABA) derivative used as a skeletal muscle relaxant.
DC9935	Basmisanil(RG1662) Featured	Basmisanil is a highly selective inverse agonist/negative allosteric modulator of α5 subunit-containing GABAA receptors which is under development by Roche for the treatment of cognitive impairment associated with Down syndrome.
DC10843	CGP 52432 Featured	CGP 52432 is a potent, selective GABAB receptor antagonist (IC50 = 85 nM).
DC12100	Cirsimaritin	Cirsimaritin binds weakly to the benzodiazepine site on GABAA receptors, with antidepressant, anxiolytic and antinociceptive activities.
DC7009	CNS-7056	CNS 7056 is a new short-acting sedative/anaesthetic that acts on GABAA receptors in the brain.
DC8706	Emamectin Benzoate	Emamectin Benzoate works as a chloride channel activator by binding gamma aminobutyric acid (GABA) receptor and glutamate-gated chloride channels disrupting nerve signals within arthropods.
DC8821	Etifoxine Hydrochloride Featured	Etifoxine Hydrochloride is a psychotropic agent with anxiolytic and anticonvulsant activity. Etifoxine Hydrochloride is an activator of GABAA R β2 and GABAA R β3.
DC11309	Fipronil	Fipronil is an insecticide that acts as a selective antagonist of insect GABA receptors (IC50s = 30 and 1,600 nM for cockroach and rat receptors, respectively).
DC9451	Flumazenil	Flumazenil(Ro 15-1788) is a benzodiazepine antagonist, non-selective for α1, α2, α3 or α5-containing GABAA receptors.
DC10158	Fluralaner Featured	Fluralaner (INN) is a systemic insecticide and acaricide Fluralaner through potent blockage of GABA and L-glutamate gated chloride channels.
DC9381	Gabapentin (hydrochloride)	Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog.
DC8954	Gabapentin Featured	Gabapentin (Neurontin) is a pharmaceutical drug, specifically a GABA analog. It was originally developed to treat epilepsy, and currently is also used to relieve neuropathic pain.
DC11090	GR3027 Featured	GR3027 (Golexanolone) is a GABA-A receptor modulating steroid antagonist that selectively antagonizes the enhanced activation of GABAA receptors by neurosteroids such as allopregnanolone and THDOC.
DC11118	HZ-166	HZ-166 (HZ166) is a GABAA receptor subtype-selective benzodiazepine site ligand with preferential activity at α2- and α3-GABA(A) receptors.
DC4137	Indiplon Featured	Indiplon is a novel sedative-hypnotic recently approved for the treatment of insomnia.
DC10853	LAU159 Featured	LAU159 is a novelα6β3γ2 GABAA receptor inhibitor.
DC8642	Lorediplon Featured	Lorediplon is a new GABAA modulator Drug for treatment of insomnia.
DCAPI1574	Nefiracetam	Nefiracetam is a nootropic of the racetam family. Nefiracetam is cognitive enhancer with an IC50 of approximately 150–200 μM for Ro 5-4864. This compound activates L/N-type calcium channels, cholinergic, monoaminergic and GABAergic systems. Nefiracetam di
DC8083	NS11394 Featured	NS11394 possesses a functional efficacy selectivity profile of alpha(5) > alpha(3) > alpha(2) > alpha(1) at GABA(A) alpha subunit-containing receptors.
DC11267	ONO-8590580 Featured	ONO-8590580 is a Novel GABAAα5 Negative Allosteric Modulator Enhances Long-Term Potentiation and Improves Cognitive Deficits in Preclinical Models.
DC10292	Pagoclone	Pagoclone is an active (+)-enantiomer of the racemate RP 59037. Pagoclone is a partial GABA(A) receptor agonist used for the treatment of panic and anxiety disorders.
DC10113	Pipequaline Featured	Pipequaline (PK 8165) is a partial benzodiazepine receptor agonist with anxiolytic activity.
DCAPI1330	Piracetam	Piracetam is a cyclic derivative of the neurotransmitter ã-aminobutyric acid (GABA), used in treatment of a wide range of cognitive disorders.
DC10578	rac BHFF Featured	Rac BHFF is a potent and selective GABAB receptor positive allosteric modulator that increases the efficacy and potency of GABA ( > 149% and > 15-fold respectively). Orally active and exhibits anxiolytic activity in vivo.

GABA Receptor

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