Home > Inhibitors & Agonists > Nuclear Receptor/Transcription Factor > Rev-ErbA
Cat. No. Product name CAS No.
DC70458 GSK-2945

GSK-2945 is a potent and selective small molecule Rev-Erbα agonist with EC50 of 50 nM, displays >1,000-fold selectivity over LXRα; inhibits LPS induction of IL-6 production and to upregulate expression of ABCA1 in human THP-1 cells; demonstrates in vivo bioavailability and orally active.

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