Novel highly selective inhibitor of multidrug resistance protein 4 (MRP4)

First-generation cephalosporin antibiotic and interleukin 15 inhibitor, specifically interacting with interleukin 15 (IL-15) receptor subunit α (IL-15Rα) and to inhibit IL-15-dependent TNF-α and IL-17 synthesis, showing inhibitory activity against all of

Third-generation, semi-synthetic, beta-lactam cephalosporin antibiotic with antibacterial activity

Second-generation, semi-synthetic, beta-lactam cephalosporin antibiotic with antibacterial activity

Broad-spectrum, beta-lactamase-resistant, second-generation cephalosporin antibiotic, inhibiting bacterial cell wall synthesis via inhibition of cross-linking of peptidoglycans

Third-generation broad spectrum antibiotic against both gram-positive and gram-negative microorganisms

Fourth-generation cephalosporin

Broad-spectrum fourth-generation cephalosporin antibiotic

beta-Lactamase-stable, broad-spectrum, third-generation cephalosporin antibiotic with antibacterial activity

Broad-spectrum, fifth-generation cephalosporin antibiotic, inactivating penicillin-binding proteins (PBPs) located on the inner membrane of the bacterial cell wall

Novel modulator of cell death signal transduction pathways, reducing the cytotoxicity of anthrax lethal toxin (LT)

Novel highly selective TAF1 inhibitor

Novel potent ALK inhibitor. also inhibiting the insulin receptor

Novel potent ALK inhibitor

Prodrug of CEP-751 (KT-6587) as antitumor agent, inhibiting protein kinases

Novel potent, selective, and orally bioavailable inverse agonist of the histamine H 3 receptor (H 3 R)

Novel selective inhibitor of the nuclear enzymes poly(ADP-ribose) polymerase (PARP) 1 and 2

Natural disrupter of RNA G-quadruplexes, inhibiting G-quadruplex-dependent alternative splicing, stimulting the stomach lining and inducing vomiting

Novel small molecule prodrug for use with SEAKER cells, exhibiting enhanced anticancer activity

Novel probe for cellulose synthase trafficking, inhibiting cellulose deposition and interferes with the trafficking of cellulose synthase complexes and their associated proteins KORRIGAN1 and POM2/CSI1

Novel Probe for the High Temperature Requirement A (HTRA) Serine Proteases

Novel non-steroid reversible dual inhibitor of CYP17 and CYP11B2 against prostate cancer with fewer cardiac side effects