Potent inhibitor of TTK kinase

Novel Highly Potent, Selective, Bioavailable TTK (threonine tyrosine kinase) Inhibitor

Novel GSK3 inhibitor, inducing cell death through cyclin D1 depletion in breast cancer cells

Novel inducer of neural differentiation and growth arrest in human primary GBM-derived cells, playing a tumor-suppressive role via cAMP/CREB signaling pathway

Novel PRL-3 inhibitor, blocking the migration and invasion of metastatic cancer cells

CGA-JK3 is CGA-JK3 is an ATP-competitive inhibitor of IKKβ-catalyzed kinase activity. CGA-JK3 inhibits IκBα phosphorylation in LPS (HY-D1056) - induced RAW 264.7 cells.

Novel functional Gboxin analogue that is suitable for live-cell ultraviolet crosslink conjugation and click chemistry

Novel Bruton's tyrosine kinase (BTK) inhibitor

Novel inhibitor of Wnt/β-catenin signaling; Anticancer agent promoting PKCα-mediated β-catenin phosphorylation/degradation

Non-peptide tachykinin NK1 receptor antagonist

Activator of RORalpha, inducing growth arrest in androgen-independent DU 145 prostate cancer cells

Novel HIV-1 protease inhibitor, also potently inhibiting major aspartyl peptidase 1 (May1), a secreted Cryptococcus neoformans protease

Peptoid Tat/transactivation response element inhibitor, inhibiting human immunodeficiency virus replication by blocking CXC-chemokine receptor 4-mediated virus entry

Liver specific thyromimetic agonist of thyroid hormone receptor-

Broad spectrum matrix metalloproteinase (MMP) inhibitor

Mutant firefly luciferase variant with enhanced light emission

Matrix metalloproteinase (MMP) inhibitor

Water soluble CycLuc3, mutant firefly luciferase variant with enhanced light emission

Benzodiazepine antagonist

Benzodiazepine receptor partial agonist

The first small-molecule based MCM2-targeted NIR-II probe

Novel Highly Potent and Selective Cholesterol 24-Hydroxylase (CH24H) Inhibitor