The first fluorogenic dipeptide probe for

Novel pan-inhibitor of sialyltransferase (ST)

Potent, selective, and orally active inhibitor of semicarbazide-sensitive amine oxidase (SSAO) activity, inhibiting vascular adhesion protein 1 (VAP-1) activity and decreasing the density of macrophages in inflamed atherosclerotic plaques in mice

Highly

Novel selective agonist of the human melanocortin 1 receptor (hMC1R) for sunless tanning and prevention of genotoxicity of UV in melanocytes

Novel inducer of biofilm dispersal, having a slower rate of NO release

Novel inhibitor of kallikrein-related peptidase 7 (KLK7) and epidermal elastase 2 (ELA2)

Novel Modulator of p75NTR-dependent motor neuron death

Negative control for LM11A-24

Novel Probe for Imaging Tau Pathology in Transgenic Mouse and Rat Models

Novel p75NTR antagonist

Novel AI-2 quorum-sensing inhibitor, affecting the starvation response and reducing virulence in several Vibrio species, most likely by interfering with LuxPQ

Novel highly selective inhibitor of the low-molecular-weight protein tyrosine phosphatase (LMPTP), being highly orally bioavailable and reversing obesity-induced diabetes in mice

Novel Two-in-One Mutant-Selective Epidermal Growth Factor Receptor Inhibitor That Spans the Orthosteric and Allosteric Sites

Potent and selective ligand of imidazoline 1 receptor (I 1 R)

Novel potent and specific agonist of I 1 imidazoline receptors

Peroxisome proliferator-activated receptor-α/γ (PPAR α/γ) dual agonist

Inhibitor of the Vesicular_monoamine_transporter_2>vesicular monoamine transporter-2 (VMAT2)

Antibiotic for treatment of bacterial infections including bronchitis and urinary tract infections, prevent urinary tract infections prior to surgery

Natural neurotrophic agent

Opioid receptor agonist, acting on the µ-opioid receptors in the myenteric plexus of the large intestine

Lopinavir Secondary Metabolite