Novel reversible monoacylglycerol lipase (MAGL) inhibitor

Inhibitor of TNF-α, preventing and restoring memory deficits associated with neuropathic pain

Inhibitor of the amebicidal activity of activated murine macrophages, helping the parasite to survive within the mouse large intestine and increasing the survival of C. elegans exposed to H2O2

Potent CB2 receptor inverse agonist

Selective modulator of plasmodial Hsp70s with antimalarial activity

Toll-like receptor 2/6 (TLR-2/6) agonist, regulating Lcn2 gene, promoting collateral growth

TLR2/6 agonist, activating the MyD88 pathway, provoking natural killer (NK) cell activation, increasing co-stimulators CD80/86 and CD40

Novel quantitative chemical probe for live cell labeling and imaging of proteins that are sensitive to redox modifications

Natural anticancer, anti-inflammatory, neuroleptic agent, also having human acyl-CoA:cholesterol acyltransferase (ACAT) inhibitory activities

Highly potent, selective, competitive, and reversible inhibitor of monoamine oxidase B (MAO-B).

Novel potent and highly selective MAO-B Inhibitor

Potent and selective MAO-B inhibitor

Novel potent selective and competitive inhibitor of MAO-B (IC 50 : 0.69 μM)

Novel potent and competitive inhibitor of MAO-B (IC 50 : 0.51 μM), also inhibiting BChE (IC 50 : 7.00 μM)

Novel selective MAO-B inhibitor

Novel stable antibody-drug conjugate (ADC) in mouse serum

Inhibitor of neuronal norepinephrine reuptake, reducing symptoms of anxiety associated with depression.

Novel highly efficient dual type I/II FMS-like tyrosine kinase inhibitor, disrupting the growth of leukemic cells

Inhibitor of voltage-gated K(+) (Kv) channels Kv1.3 and Kv1.5

Novel, active, and less toxic anti-tuberculosis (anti-TB) agent

Neurokinin receptor antagonist with antiemetic activity

Novel potent tyrosinase inhibitor from the Gram-negative bacterium Massilia albidiflava DSM 17472T