Blocker of dsRNA-induced IRF3 nuclear translocation and homodimerization; Inhibitor of lipopolysaccharide-mediated Toll-like receptor-4 signaling; Inhibitor of human pancreatic cancer

Novel selective α-syn ligand, exhibited the promising binding characteristics for α-syn aggregates (Ki = 0.52 nM)

Novel neuropeptide, protecting human brain vascular endothelial cells against oxygen-glucose deprivation/reoxygenation (OGD/R)-induced inflammation and permeability, significantly ameliorating HFD-induced obesity and fatty liver, regulating pituitary gona

Novel GPR173 agonist, promoting osteoblastic differentiation of MC3T3-E1 cells. stimulating mRNAs encoding hypothalamo-pituitary-gonadal hormones

Natural anti-tumor agent, showing strong apoptotic anticancer effects against platinum-resistant solid cancers

Potent antagonist of (H1N1)pdm09 infection, markedly suppressing cytopathic effects and attenuating viral gene expression in (H1N1)pdm09-infected MDCK cells

Sulindac derivative with promising anticancer activities

Inducer of platelet aggregation, playing a role in cellular signal transduction and possibly in cell growth control and carcinogenesis

Novel photoswitchable BET bromodomain Degrader (PHOTAC)

Novel potent photoswitchable antagonist for a precise spatiotemporal control of β2-adrenoceptors

Novel photocontrol inhibitor of the voltage-gated proton channel Hv1

Functionalized photoswitchable cereblon ligand for Degraders

Novel photoswitchable sphingolipid probe, reversibly controlled S1P3-dependent pain hypersensitivity in mice and uniquely suited for the study of S1P biology in cultured cells and in vivo

Novel porphyrazine-based photodynamic anti-cancer agent, inducing immunogenic cell death

Novel porphyrazine-based photodynamic anti-cancer agent, inducing immunogenic cell death

Novel photoswitchable sphingolipid probe

Novel photoswitchable inhibitor of human dihydrofolate reductase

Natural flavonoidal alkaloid from the sea-grass Phyllosphadix iwatensis

Natural cytotoxic withanolide antitumor agent, inducing apoptosis by decreasing mitochondrial membrane potential and elevating the Bax/Bcl-2 protein expression ratio

Natural inhibitor of Wnt signaling, modulating β-catenin-dependent transcription

Platelet aggregation inhibitor

Platelet aggregation inhibitor