Novel Human Toll-like Receptor 8-Selective Agonist

Stimulator of metabolism, preventing diseases associated with parturition and peri-partum period, developmental and nutritional disorders in young animals, and bone growth disorders and tetany or paresis caused by calcium, magnesium, and phosphorus metabo

Natural agonist of TPRC1/4/5 channels, also acting as a dual PKCα and PKCθ activator, inducing an insulin resistant phenotype by inhibiting IRS1 and the PI3K/Akt pathway, activating the heat shock factor 1 (HSF1) transcription factor driving glucose depen

Novel dual TOP1 and TDP1 inhibitor, inducing both cellular TOP1cc, TDP1cc formation and DNA damage, resulting in cancer cell apoptosis at a sub-micromolar concentration

Novel narrow spectrum kinase inhibitor, potently inhibiting P38a, Src, and Syk kinase activities

Novel Selective Inhibitor of Endoplasmic Reticulum α-Glucosidase II, Exhibiting Antiflaviviral Activity

Novel highly specific fluorescent TOPK inhibitor

Nucleic acid stain, acting on viable, early apoptotic and necrotic cells differentially, showing specific staining of nuclei without any staining of the cytoplasm

Natural psychoactive agent

Chromogenic peptide substrate for the rapid and specific photometric assay of recombinant hirudin (r-hirudin)

Selective CA IX inhibitor

Novel ToxT inhibitor, reducing Vibrio cholerae virulence in vivo and effectively inhibiting intestinal colonization in the infant mouse

Novel probe for activin receptor-like kinase (ALK4 and ALK5)

Novel inhibitor of O-GlcNAcase (OGA)

Novel probe for CECR2/BPTF bromodomains

First-in-class fluorescent drug delivery vesicle that can efficiently load both water-soluble and -insoluble anticancer drugs

Novel Peripheral Selective Tryptophan Hydroxylase 1 (TPH1) Inhibitor (IC 50 : 42nM) for Obesity and Fatty Liver Disease

Inhibitor of tyrosine recombinases and Holliday junction-resolving enzymes; Antibacterial

Promising amyloid reducing agent by lowering the levels of Aβ.

Novel Specific Inhibitor of Type I Collagen Production in Fibrosis

Novel taxane family member, reducing the brain metastatic colonization of breast cancer cells

Novel tumour progression locus 2 (Tpl2) kinase inhibitor