Cat. No. | Product name | CAS No. |
DC23955 |
PF-04929113 Mesylate
The prodrug of PF-04928473 (SNX-2112), a potent, orally bioavailable HSP90 inhibitor. |
1173111-67-5 |
DC23989 |
TG 100801 hydrochloride
The prodrug of TG 100572, a potent, dual receptor tyrosine kinase/Src kinase inhibitor with IC50 of 2-16 nM for VEGFR, FGFR and PDGFR, 0.1-5 nM for Src family. |
1018069-81-2 |
DC22456 |
GLPG-0492 R enantiomer
The R enantiomer of GLPG-0492, a non-steroidal selective androgen receptor modulator (SARM) for treatment for Duchenne muscular dystrophy (DMD). |
1215085-93-0 |
DC24174 |
Refametinib R enantiomer
The R enantiomer of Refametinib, a potent, non–ATP-competitive, highly selective, allosteric inhibitor of MEK1/2 with IC50 of 19/47 nM respectively.. |
923032-38-6 |
DC24133 |
Bay 65-1942 R form
The R form of Bay 65-1942. which is a potent, selective, ATP-competitive inhibitor of IKKβ kinase with Ki of 2 nM.. |
758683-21-5 |
DC23865 |
LOXO-195 R racemate
The R racemate of LOXO-195, a potent, selective, next-generation Trk tyrosine kinase inhibitor with IC50 of 0.6 nM and <2.5 nM for WT TrkA and WT TrKC, respectively.. |
1350884-56-8 |
DC23174 |
GNE-140 racemate
Featured
The racemate of GNE-140, a novel potent, selective lactate dehydrogenase (LDH) inhibitor with IC50 of 3, 5, and 5 nM for LDHA, LDHB, and LDHC, respectively. |
1802977-61-2 |
DC22558 |
Pemafibrate racemate
The racemate of Pemafibrate, which is a highly potent, specific PPARα agonist with EC50 of 1 nM.. |
848258-31-1 |
DC23999 |
(R)-Oxiracetam
the R-enantiomer of the nootropic drug oxiracetam (ISF 2522), which is a nootropic drug of the racetam family and stimulant.. |
68252-28-8 |
DC23866 |
LOXO-195 RS-isomer
The RS-isomer of LOXO-195, a potent, selective, next-generation Trk tyrosine kinase inhibitor with IC50 of 0.6 nM and <2.5 nM for WT TrkA and WT TrKC, respectively.. |
2097002-59-8 |
DC22480 |
5-FAM
The single isomer, 5-FAM, contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid. Fluorescein is the most common fluorescent derivatization reagent for labeling biomolecules. In addition |
76823-03-5 |
DC9377 |
6-FAM
The single isomer, 6-FAM, contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid. |
3301-79-9 |
DC20816 |
BMS 830216
The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM. |
1197420-06-6 |
DC11492 |
GMX-1777 chloride
The water-soluble prodrug of GMX-1778 (CHS-828), which is a potent and specific inhibitor of the NAD(+) biosynthesis enzyme NAMPT with IC50 of <20 nM. |
432037-57-5 |
DC22593 |
KPT-8602 Z-isomer
The Z-isomer of Eltanexor (KPT-8602), which is a second-generation SINE with markedly reduced brain penetration compared to selinexor.. |
1642300-78-4 |
DC22541 |
R-80123
The Z-isomer of R 79595, a highly selective PDE inhibitor, 10-fold more potent than R 79595.. |
133718-30-6 |
DC20173 |
Acefylline;Theophyllineacetic acid; Theophylline-7-acetic acid
Theophylline-7-acetic acid (Acefylline), acting as an adenosine receptor antagonist, is a stimulant drug of the xanthine chemical class. |
652-37-9 |
DC8759 |
Thiamet G
Featured
Thiamet G is a potent and selective inhibitor of O-GlcNAcase that demonstrates a Ki value of 21 nM. |
1009816-48-1 |
DC8673 |
Thifluzamide
Thifluzamide is a powerful and effective fungicide. When used safely and correctly it can be effective on rice and other crops because of improved water dispersal techniques. Thifluzamide is highly active against Basidiomycete fungi, in particular Rhizoct |
130000-40-7 |
DC12363 |
Thionin acetate (Thionine acetate)
Thionin (acetate) is a metachromic cationic histology dye used in biological staining widely. |
78338-22-4 |
DC11362 |
Thiothixene
Thiothixene is a typical antipsychotic.1 It selectively binds to dopamine D2 over D1, D3, and D4 receptors (Kis = 0.417, 338, 186.2, and 363.1 nM, respectively). |
5591-45-7 |
DC12573 |
THIQ40
THIQ 40 (THIQ40) is a potent, orally available ERα antagonist and selective estrogen receptor degrader (SERD) with IC50 of 17 nM (ERα binding) and 30 nM (ERα transcription), IC50 of 0.9 nM (ERα degradation). |
1799430-91-3 |