Home > Products > Novel inhibitors
Cat. No. Product name CAS No.
DC23955 PF-04929113 Mesylate

The prodrug of PF-04928473 (SNX-2112), a potent, orally bioavailable HSP90 inhibitor.

1173111-67-5
DC23989 TG 100801 hydrochloride

The prodrug of TG 100572, a potent, dual receptor tyrosine kinase/Src kinase inhibitor with IC50 of 2-16 nM for VEGFR, FGFR and PDGFR, 0.1-5 nM for Src family.

1018069-81-2
DC22456 GLPG-0492 R enantiomer

The R enantiomer of GLPG-0492, a non-steroidal selective androgen receptor modulator (SARM) for treatment for Duchenne muscular dystrophy (DMD).

1215085-93-0
DC24174 Refametinib R enantiomer

The R enantiomer of Refametinib, a potent, non–ATP-competitive, highly selective, allosteric inhibitor of MEK1/2 with IC50 of 19/47 nM respectively..

923032-38-6
DC24133 Bay 65-1942 R form

The R form of Bay 65-1942. which is a potent, selective, ATP-competitive inhibitor of IKKβ kinase with Ki of 2 nM..

758683-21-5
DC23865 LOXO-195 R racemate

The R racemate of LOXO-195, a potent, selective, next-generation Trk tyrosine kinase inhibitor with IC50 of 0.6 nM and <2.5 nM for WT TrkA and WT TrKC, respectively..

1350884-56-8
DC23174 GNE-140 racemate Featured

The racemate of GNE-140, a novel potent, selective lactate dehydrogenase (LDH) inhibitor with IC50 of 3, 5, and 5 nM for LDHA, LDHB, and LDHC, respectively.

1802977-61-2
DC22558 Pemafibrate racemate

The racemate of Pemafibrate, which is a highly potent, specific PPARα agonist with EC50 of 1 nM..

848258-31-1
DC23999 (R)-Oxiracetam

the R-enantiomer of the nootropic drug oxiracetam (ISF 2522), which is a nootropic drug of the racetam family and stimulant..

68252-28-8
DC23866 LOXO-195 RS-isomer

The RS-isomer of LOXO-195, a potent, selective, next-generation Trk tyrosine kinase inhibitor with IC50 of 0.6 nM and <2.5 nM for WT TrkA and WT TrKC, respectively..

2097002-59-8
DC22480 5-FAM

The single isomer, 5-FAM, contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid. Fluorescein is the most common fluorescent derivatization reagent for labeling biomolecules. In addition

76823-03-5
DC9377 6-FAM

The single isomer, 6-FAM, contains a carboxylic acid that can be used to react with primary amines via carbodiimide activation of the carboxylic acid.

3301-79-9
DC20816 BMS 830216

The the phosphate ester prodrug of BMS 819881, a potent, selective melanin concentrating hormone receptor 1 (MCHR1) inhibitor with Ki of 10.4 nM.

1197420-06-6
DC11492 GMX-1777 chloride

The water-soluble prodrug of GMX-1778 (CHS-828), which is a potent and specific inhibitor of the NAD(+) biosynthesis enzyme NAMPT with IC50 of <20 nM.

432037-57-5
DC22593 KPT-8602 Z-isomer

The Z-isomer of Eltanexor (KPT-8602), which is a second-generation SINE with markedly reduced brain penetration compared to selinexor..

1642300-78-4
DC22541 R-80123

The Z-isomer of R 79595, a highly selective PDE inhibitor, 10-fold more potent than R 79595..

133718-30-6
DC20173 Acefylline;Theophyllineacetic acid; Theophylline-7-acetic acid

Theophylline-7-acetic acid (Acefylline), acting as an adenosine receptor antagonist, is a stimulant drug of the xanthine chemical class.

652-37-9
DC8759 Thiamet G Featured

Thiamet G is a potent and selective inhibitor of O-GlcNAcase that demonstrates a Ki value of 21 nM.

1009816-48-1
DC8673 Thifluzamide

Thifluzamide is a powerful and effective fungicide. When used safely and correctly it can be effective on rice and other crops because of improved water dispersal techniques. Thifluzamide is highly active against Basidiomycete fungi, in particular Rhizoct

130000-40-7
DC12363 Thionin acetate (Thionine acetate)

Thionin (acetate) is a metachromic cationic histology dye used in biological staining widely.

78338-22-4
DC11362 Thiothixene

Thiothixene is a typical antipsychotic.1 It selectively binds to dopamine D2 over D1, D3, and D4 receptors (Kis = 0.417, 338, 186.2, and 363.1 nM, respectively).

5591-45-7
DC12573 THIQ40

THIQ 40 (THIQ40) is a potent, orally available ERα antagonist and selective estrogen receptor degrader (SERD) with IC50 of 17 nM (ERα binding) and 30 nM (ERα transcription), IC50 of 0.9 nM (ERα degradation).

1799430-91-3
Page 262 / Total 1557 FirstPrevNextLastGoto