Firefly luciferin analog as a key element of bioluminescent reporters for oxidation state and thiol/disulfide equilibria

GABAA receptor agonist

Novel Potent Inhibitor of the Opioid Receptors and the Ion Channels

Novel inducer of apoptotic cell death in platinum-resistant A2780cis human ovarian cancer cells, exhibitong a strong inhibitory effect in ovarian CSC-LCs in combination with cisplatin

Steroidomimetic and Chimeric Microtubule Disruptor

Selective Tau ligand, selectively binding to neurofibrillary tangles and neuropils in people with Alzheimer's disease

Novel orthosteric-allosteric dual inhibitor of PfHT1 as selective antimalarial agent

Novel orthosteric-allosteric dual inhibitor of PfHT1 as selective antimalarial agent

Novel orthosteric-allosteric dual inhibitor of PfHT1 as selective antimalarial agent

Novel potent, highly selective and orally available PI3Kδ inhibitor

Novel phosphodiesterase 10A (PDE10A) inhibitor for treatment of schizophrenia

Phosphodiesterase 10A (PDE10A) inhibitor

Novel dose-dependent inhibitor of HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, and HDAC9; NOX Inhibitor

Novel selective thrombin inhibitor, inducing conformational allostery

Novel multivalent ligand that bridges the allosteric and orthosteric binding sites of the M2 muscarinic receptor

Anti-epileptic and anticonvulsant agent, acting as a selective GABA reuptake inhibitor

Anthraquinone-fused enediyne antitumor agent for development of antibody-drug conjugates (ADCs)

Muscarinic receptor antagonist, anticholinergic,and parasympatholytic

Natural anticancer agent fortreatment of mast cell tumor (MCT)

Widely used oxidation-reduction indicator

Macrolide antibiotic for the treatment of bovine respiratory disease and ovine respiratory disease associated with Mannheimia (Pasteurella) haemolytica

Antiviral, antineoplastic, and anti-inflammatory agent; Orally active interferon inducer, inhibiting Ebola virus (EBOV)