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Cat. No. Product name CAS No.
DCC5462 Vu0477886

Novel potent mGlu4 PAM with an attractive DMPK profile, and robust efficacy in preclinical Parkinsons disease model, haloperidol-induced catalepsy (HIC)

DCC5463 Vu0486321

mGlu1 positive allosteric modulator (PAM)

1816301-67-3
DCC5464 Vu0487836

Novel cyclooxygenase-1 (COX-1)-selective inhibitor

1632301-78-0
DCC5465 vu573 Hydrochloride

Novel modulator of mammalian inward rectifying potassium (Kir) channels

1049717-96-5
DCC5466 Vu6001192

Novel selective negative allosteric modulator (NAM) of metabotropic glutamate receptor subtype 2

1821325-29-4
DCC5467 Vu6004909

Novel potent and highly selective mGlu1 PAM (22nM), reducing striatal DA release in vivo and displaying antipsychotic efficacy

DCC5468 Vu6007705

Novel Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM)

2222737-18-8
DCC5469 Vu6008555

Novel Muscarinic Acetylcholine Receptor Positive Allosteric Modulator (PAM)

2222737-14-4
DCC5470 Vu6009453

Novel M4 positive allosteric modulator (PAM)

2148929-11-5
DCC5471 Vu6009833

Novel CNS penetrant pan-muscarinic antagonist

DCC5472 Vu6013429

Novel PAM of Group III (mGlu4/6/7/8) mGlu receptors

DCC5473 Vu6017587

Novel selective mGlu3 NAM, showing efficacy in tail suspension, elevating zero maze and marble burying, suggesting selective inhibition of mGlu3 affords anxiolytic-like and antidepressant-like phenotypes in mice

DCC5474 Vu6027459

First-in-class selective mGlu7 positive allosteric modulator (PAM), displaying CNS penetration in both mice (Kp = 2.74) and rats (Kp= 4.78)

DCC5475 Vuf 5681 Dihydrobromide

Potent histamine H3 receptor silent antagonist

639089-06-8
DCC5476 Vuf10132

Novel full inverse agonist at CXCR3 N3.35A

1037732-88-9
DCC5477 vuf10148

Potent H4R ligand

1001065-53-7
DCC5478 Vuf10166 Hydrochloride

Novel potent ligand at 5-HT3A and 5-HT3AB receptors with different activities

55686-37-8
DCC5479 Vuf10497 Featured

VUF10497 is a potent histamine H4 receptor (H4R) inverse agonist with anti-inflammatory activity.

1080623-12-6
DCC5480 Vuf10499

Potent human H4 receptor inverse agonist

1080623-05-7
DCC5481 Vuf10558

Highly Potent Human Histamine H4 Receptor Inverse Agonist

1166378-39-7
DCC5482 Vuf11211

Potent CXCR3 Antagonist, extending from the minor pocket into the major pocket of the transmembrane domains and binding between residues in helices 1 (Y1.39), 2 (W2.60), 3 (F3.32), 4 (D4.60), 6 (Y6.51), and 7 (S7.39, Y7.43)

906556-51-2
DCC5483 Vuf11222

First reported nonpeptidomimetic agonist on The G protein-coupled chemokine receptor CXCR3

1414376-84-3
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