Cat. No. | Product name | CAS No. |
DC74428 |
Adrixetinib
Adrixetinib is a small molecule inhibitor of Axl/Mer RTK. |
2394874-66-7 |
DC74429 |
ER-851
ER851 (ER-851) is a potent and highly selective AXL inhibitor. |
|
DC74430 |
INCB081776
INCB081776 is a potent and selective dual inhibitor of AXL and MERTK with IC50 of 16 and 14 nM respectively, 30-fold selectivity over TYRO3. |
|
DC74431 |
R992
R992 (MERTK inhibitor) is a novel potent, selective and orally bioavailable inhibitor of Mer tyrosine kinase (MerTK) with IC50 of 18 nM in ADP-Glo assays. |
2171523-99-0 |
DC74432 |
UNC2025 hydrochloride
UNC2025 is a potent, orally bioavailable Mer/FLT3 dual inhibitor with IC50 of 0.74/0.8 nM, 700-fold less active against Met compared to Mer. |