Antioxidant, free radical scavenger and potent inhibitor of lipid peroxidation

Mixture of Meropenem and vaborbactam for adults with complicated urinary tract infections (cUTI), including a type of kidney infection, pyelonephritis, caused by specific bacteria

Analog of etomidate that interacts weakly with 11β-hydroxylase

Novel fluorescent probe targeting of G-quadruplex structures and trapping cytoplasmic RNA G-quadruplex structures in cells

Inducer of deformation in Zebrafish>Zebrafish through the AhR-mediated, CYP1A-independent pathway

Novel inhibitor of full-length GST-tagged CARM-1

Novel potent inhibitor of coactivator-associated arginine methyltransferase 1 (CARM1)

Novel, potent, long-acting, selective, orally bioavailable inhibitor of dipeptidyl peptidase 4 (DPP-4) with hypoglycemic activity

Anthracycline antineoplastic antibiotic, intercalating into DNA and interacting with topoisomerase II, thereby inhibiting DNA replication and repair and RNA and protein synthesis.

Long acting ß2-adrenoreceptor agonist (LABA)

Novel orally available α4 integrin receptor inhibitor

Irreversible and nonselective Monoamine_oxidase_inhibitor>monoamine oxidase inhibitor (MAOI)

DNA minor groove alkylating agent, alkylating N3 of adenine in a consensus sequence 5'-(A/T)(A/T)A*

Novel Cas9 Inhibitor, direct binding to apo-Cas9, preventing Cas9:gRNA complex formation

The first inhibitor of fungal (1→3)-β-D-glucan synthesis

Natural potent neutrophil elastase (NE) inhibitor with an IC 50 value of 2.79 ± 0.07 μM

Novel activator of autophagy for potential treatment of cystic fibrosis

Selective inhibitor of cathepsin B endopeptidase and exopeptidase activities

Selective inhibitor of cathepsin B endopeptidase and exopeptidase activities

Novel selective reversible inhibitor of cathepsin X

Novel ligand of voltage-gated calcium channel α2δ-1 subunit (Cavα2δ-1)

Selective inhibitor of 15-hydroxy PGDH, significantly suppressing endogenous 11-oxo-ETE production with a corresponding increase in 11(R)-HETE