Isoform-selective inhibitor of histone deacetylase (HDAC1)

Novel potent CysLT2 receptor antagonist

Novel Mdm2 inhibitor, an analog of Nutlin-3

Novel Mdm2 inhibitor, an analog of Nutlin-3

Novel RAF kinase inhibitor

Novel SRC kinase inhibitor

Novel IκB kinase inhibitor

Novel Thymidine kinase (TK) inhibitor

Novel Cyclin-dependent kinase inhibitor

Novel IκB kinase inhibitor

Novel Cell_cycle>cell cycle inhibitor

Dual thymidylate synthase and dihydrofolate reductase inhibitor

Novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro

Selective sphingosine kinase 1 (SK1) inhibitor

Novel inhibitor of HIV-1 entry

Novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro

Selective inhibitor of Adenylyl Cyclase isoform-2 (AC2)

Novel inhibitor of HIV-1 gene expression

Novel potent inhibitor of filamentation and biofilm formation by the Candida albicans SC5314 strain

Novel inhibitor of Mycobacterium marinum MelF (Rv1936), exhibiting bacteriostatic/bactericidal activity against M. marinum and M. tuberculosis in vitro

Novel Protein kinase A and B inhibitor

The first clickable, photoreactive probe that inhibits both γ-secretase and PSase activities and specifically labels PS1-NTF and signal peptide peptidase (SPP)