Selective inhibitor of hCA IX and hCA XII

Potent and selective inhibitor of cathepsin B

Novel specific inhibitor of cathepsin L, effectively inhibiting degradation of LC3-II and GABARAP

Novel selective CaBdf1 BD1 inhibitor

Novel inhibitor of CaBdf1 BD1 with low-micromolar affinity and three- to fivefold selectivity relative to human Brd4 BD1

Novel selective CaBdf1 BD2 inhibitor

Potent, selective class B inhibitor of calcium-activated chloride channels (CaCCs)

Novel photocaged ERK1/2 inhibitor as a light-controlled anticancer agent

Potent agonist at thyroid hormone receptor (TR)

Effective inhibitor of the carbonic anhydrase (CA) from Trypanosoma cruzi (TcCA)

Novel inhibitor of p110

Cell permeable derivative of calcein, becoming fluorescent on hydrolysis

Dual inhibitor of fibroblast growth factors (FGF) and vascular endothelial growth factor (VEGF) ; Anti-angiogenic

Ionophore highly selective for Ca , potentiating responses to NMDA but not quisqualate

Transmembrane protease serine 2 (TMPRSS2) inhibitor for the treatment of chronic pancreatitis and postoperative gastric reflux, blocking SARS-CoV-2 replication in TMPRSS2-expressing human cells

Novel destabilizer of CAND1-Cullin1 interaction, inducing a p53-stress response pathway

Natural cannabinoid precursor

Natural cannabinoid precursor

Novel self-assembling lysine-rich cationic amphipathic peptide (CAP)

Reverse-transcriptase_inhibitor>Non-nucleoside reverse transcriptase inhibitor

Broad spectrum antibiotic used in the therapy of drug resistant tuberculosis as a second line agent

Antimuscarinic and anticholinergic, acting as an antagonist of NMDA receptor