Herbicide safener that is added to various herbicide formulations to reduce crop damage

Long-acting benzodiazepine, producing the active metabolite desmethyl-diazepam, which is a partial agonist of the GABAA receptor

Full agonist of GABAA receptors, acting as anxiolytic, sedative, hypnotic, amnesic, anticonvulsant and muscle relaxant agent

Precursor for tumor selective PET imaging (124I-CLR1404) or therapeutic radiation (131I-CLR1404)

Novel chromophore-linked metallo-β-lactamase (MBL) substrate as potential inhibitor against a panel of clinically relevant MBLs

Novel inhibitor of

Novel potent and selective dual inhibitor of c-Met and ALK, potently abrogating hepatocyte growth factor (HGF)-induced c-Met phosphorylation and cell migration, phosphorylation of ALK, EML4-ALK, and ALK resistance mutants in transfected cells

Novel selective agonist of cannabinoid CB2 receptors

Novel Matrix Metalloproteinase Inhibitor As a Potent Antihemorrhagic Agent

First-in-class dual PDE5 and HDAC6-selective inhibitor

Novel Epigenetic Inhibitor Targeting Histone Deacetylases, DNA Methyltransferase 1, and Lysine Methyltransferase G9a with In Vivo Efficacy in Multiple Myeloma

Novel inhibitor of

Novel Hedgehog pathway inhibitor, revealing the receptor GPR39

Novel Potent and Specific Target Of Rapamycin Complex 2 (TORC2) Inhibitor

Novel ultrapotent and selective inhibitor of of human β-Factor XIIa

Novel peptide STAT5 inhibitor, blocking IL-2/sIL-2Rα signaling and inhibiting T reg cell development

Novel SARS-CoV Mpro inhibitor which has its P1-phenylalanine residue bound to the relatively hydrophilic S1 pocket of the enzyme and yet exhibits a high inhibitory activity against SARS-CoV Mpro, with Ki = 2.24 ± 0.58 μM

Potent dual 5-lipoxygenase (5-LOX) inhibitor and platelet-activating factor (PAF) receptor antagonist

Inhibitor of DprE1, an epimerase required for cell wall biosynthesis

Novel allosteric modulator of the β2 adrenergic receptor (β2AR), binding to a pocket formed primarily by the cytoplasmic ends of transmembrane segments 1, 2, 6 and 7 as well as intracellular loop 1 and helix 8

Selective and potent potentiator of nAChRs containing an α4

Novel TRPV1 modulator, also modulating both CB1 and CB2 receptors