Highly potent, selective, competitive, and reversible inhibitor of monoamine oxidase B (MAO-B)

Novel potent Lp1NTPDase inhibitor

Novel Potent and Selective Antagonist for the UTP-Activated P2Y4 Receptor

Novel Potent Agonist of the Orphan G Protein-Coupled Receptor GPR17 (EC 50 12 nM)

Novel potent and selective agonist of the orphan G protein-coupled receptor 84 (GPR84)

Fluorescent Probe for Ecto-5'--nucleotidase (CD73)

Novel Potent Agonist of the Orphan G Protein-Coupled Receptor GPR17 (EC 50 27.9 nM)

Novel Potent Agonist of the Orphan G Protein-Coupled Receptor GPR17 (EC 50 32.1 nM)

Fluorescent Probe for Ecto-5'--nucleotidase (CD73)

The first potent and selective inhibitor of human nucleoside triphosphate diphosphohydrolase-2 (NTPDase2)

Novel Agonist of the Cannabinoid-Activated Orphan G-Protein-Coupled Receptor GPR18, being selective versus the CB-sensitive receptors CB1, CB2, and GPR55

Novel Agonist of the Cannabinoid-Activated Orphan G-Protein-Coupled Receptor GPR18, being selective versus the CB-sensitive receptors CB1, CB2, and GPR55

Potent GPR55 antagonist

Novel Selective, competitive GPR55 antagonist

Novel Highly Sensitive PSMA Probe for NIR-II Imaging and Intraoperative Tumor Resection, Visualizing Tumors in Real Time

Novel PSMA ligand conjugated with fluorescent dye SulfoCy7, demonstrating good visualization of PSMA-expressing tumors and the absence of any explicit toxicity up to 87.9 mg/kg

Na-K ATPase inhibitor, stimulating SERCA2a and accelerating calcium cycling in heart failure by relieving phospholamban inhibition

Novel Bovine Viral Diarrhea (BVD) Inhibitor, specifically blocking BVDV cell entry

Novel inhibitor of hypoxia-induced VEGF expression

Natural antifungal agent, against postharvest fruit pathogenic fungi

Novel CFTR modulator, increasing CFTR protein expression across different mutations, including F508del, by increasing CFTR mRNA levels by ~1.5 to ~2-fold in HBE cells

Novel CFTR modulator, binding to the poly-r(C) binding protein 1 (PCBP1), showing an affinity for RNA-bound PCBP1 higher than that of free PCBP1