Novel allosteric RORγt inverse agonist

Selective inhibitor of the dopamine transporter (DAT), blocking cocaine-induced locomotor stimulation and acting as a positive allosteric modulator of the human CB1 (hCB1) receptor

Novel potent and selective KOR antagonist

Novel Potent and Selective Orexin-1 Receptor Antagonist

Novel Potent Dual Orexin Receptor Agonist

Novel allosteric inhibitor of soluble adenylyl cyclase (sAC)

Potent serotonin SR-1A/SR-1B and moderate SR-2C agonist

Potent vertebrate GABAa antagonist

Novel non-steroidal antiandrogen, downregulating c-myc messenger RNAs

Potent non-steroidal antiandrogen

Novel DNA gyrase B inhibitor

Novel inhibitor of Src protein tyrosine kinase SH2

PKCβ-selective inhibitor

The first small molecule inhibitor of ThiD; IkB kinase (IKK) inhibitor; antibiotic

Novel Ricin Inhibitor, Targeting Ribosome Binding

Novel Ricin Inhibitor, Targeting Ribosome Binding

Novel Ricin Inhibitor, Targeting Ribosome Binding

Novel Ricin Inhibitor, Targeting Ribosome Binding

Inhibitor of Adipogenesis/Lipogenesis with AMPK Activation and UPR Suppression, Reducing Lipid Accumulation in Adipocytes

Novel specific RUVBL1/2 ATPase inhibitor, radiosensitizing NSCLC, but not normal lung epithelial cells

Natural potent macrophage uptake enhancer of S. aureus and zymosan A bioparticles

Inhibitor of LFA-1/ICAM-1 Mediated Cell Adhesion