Natural antibiotic, being active against P. aeruginosa both in vitro and in vivo.

Novel glutaminase activity inhibitor, showing a partial uncompetitive inhibition in vitro and a significant reduction of ammonia and glutamate production in vivo

Prodrug of Thiamphenicol, inhibiting the 50S subunit of the bacterial ribosome and protein translation

Novel antibiofilm agent, disturbing symbiotic balance between C. albicans and S. mutans in dual species biofilm

Highly efficient bioregulator of plant morphogenesis in the tissue culture technique, inducing diverse responses ranging from induction of callus to embryogenesis or organogenesis, acting through modulation of the endogenous plant growth regulators, modif

Novel protein-protein interaction inhibitor of PAC3 homodimer

Novel selective anticancer agent, selectively inducing cancer cell death in a caspase independent pathway

First-in-class potent, selective, reversible, and tight binding inhibitor of human monoamine oxidase B (hMAO-B) (hMAO-B IC 50 = 1.52 ± 0.15 nM)

Novel potent DENV2-NS2B/NS3pro inhibitor

Firefly luciferin analog as a key element of bioluminescent reporters for oxidation state and thiol/disulfide equilibria

GABAA receptor agonist

Novel Potent Inhibitor of the Opioid Receptors and the Ion Channels

Novel inducer of apoptotic cell death in platinum-resistant A2780cis human ovarian cancer cells, exhibitong a strong inhibitory effect in ovarian CSC-LCs in combination with cisplatin

Steroidomimetic and Chimeric Microtubule Disruptor

Selective Tau ligand, selectively binding to neurofibrillary tangles and neuropils in people with Alzheimer's disease

Novel orthosteric-allosteric dual inhibitor of PfHT1 as selective antimalarial agent

Novel orthosteric-allosteric dual inhibitor of PfHT1 as selective antimalarial agent

Novel orthosteric-allosteric dual inhibitor of PfHT1 as selective antimalarial agent

Novel potent, highly selective and orally available PI3Kδ inhibitor

Novel phosphodiesterase 10A (PDE10A) inhibitor for treatment of schizophrenia

Phosphodiesterase 10A (PDE10A) inhibitor

Novel dose-dependent inhibitor of HDAC1, HDAC3, HDAC4, HDAC5, HDAC6, HDAC7, HDAC8, and HDAC9; NOX Inhibitor