Chromogenic peptide substrate for the rapid and specific photometric assay of recombinant hirudin (r-hirudin)

Selective CA IX inhibitor

Novel ToxT inhibitor, reducing Vibrio cholerae virulence in vivo and effectively inhibiting intestinal colonization in the infant mouse

Novel probe for activin receptor-like kinase (ALK4 and ALK5)

Novel inhibitor of O-GlcNAcase (OGA)

Novel probe for CECR2/BPTF bromodomains

First-in-class fluorescent drug delivery vesicle that can efficiently load both water-soluble and -insoluble anticancer drugs

Novel Peripheral Selective Tryptophan Hydroxylase 1 (TPH1) Inhibitor (IC 50 : 42nM) for Obesity and Fatty Liver Disease

Inhibitor of tyrosine recombinases and Holliday junction-resolving enzymes; Antibacterial

Promising amyloid reducing agent by lowering the levels of Aβ.

Novel Specific Inhibitor of Type I Collagen Production in Fibrosis

Novel taxane family member, reducing the brain metastatic colonization of breast cancer cells

Novel tumour progression locus 2 (Tpl2) kinase inhibitor

Enhancer of the cytotoxic effect of immunotoxins (ITs) which results in increased apoptosis in different cancer cells

Mitochondria-activatable luciferin (MAL-Probe)

Novel Type-I Inhibitor of TIE-2

Potent I 2 -imidazoline receptor agonist

Metabolite of Resveratrol

Potent and selective NMDA agonist

Novel HuR binder, modulating HuR-RNA interactions

Novel KGA allosteric inhibitor

Natural resveratrol trimer, acting as a protein kinase C inhibitor