Neutral, nonandrogenic, progesterone-like profile progestin

Novel human epidermal growth factor receptor-2 (HER2) inhibitor; Spermatocide

Novel red-light-controllable nitric oxide (NO) releaser

FAUC-365 analog

Steroidal progestin used in veterinary medicine to control estrus and ovulation in cattle

Secondary metabolite from the myxobacterium Sorangium cellulosum, acting as a potent HCV inhibitor, Ebola virus (EBOV) entry inhibitor, and a potassium channel inhibitor

Controllable nitric oxide (NO) donor, releasing NO triggered by photoinduced electron transfer (PeT)

Natueal sigma receptor agonist, attenuating cytokine release associated with SARS-CoV-2, also being used as anti-malarial, anti-stroke and cough-suppressant

Novel potent inhibitor of notum carboxylesterase activity

Novel potent notum inhibitor (OPTS IC50 3.6nM; TCF-LEF EC50 220nM), showing good plasma exposure and reasonable CNS penetration

Novel potent LRRK2 inhibitor

Natural inhibitor of the allosteric regulation of Hsp70

Natural inhibitor of jasmonate signaling targets JAR1 in Arabidopsis thaliana

Second-Generation RET/VEGFR2 Inhibitor

Novel stabilizer of long noncoding RNA (lncRNA) GAS5, binding to GAS5 with high affinity, and increasing GAS5 levels and glucose uptake in diabetic patient adipocytes

Novel Inhibitor of Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1)

Novel Inhibitor of Trypanosoma brucei Phosphodiesterase B1 (TbrPDEB1)

Novel inhibitor of Trypanosoma brucei PDEB1 (TbrPDEB1)

Novel selective SIRT2 inhibitor, creating a hydrophobic cavity behind the substrate-binding pocket after a conformational change of the Zn-binding small domain of SIRT2

Novel activator of 15-ADON production, significantly increasing the transcription of Tri6, a transcription factor gene necessary for trichothecene biosynthesis, in both trichothecene-inducing and noninducing culture conditions

Novel biomediator, inducing reveromycin production in Streptomyces sp. SN-593

Novel tubulin inhibitor