| Cat. No. | Product Name | Field of Application | Chemical Structure |
|---|---|---|---|
| DC22620 | Tiadinil | A plant activator of systemic acquired resistance, boosts the production of herbivore-induced plant volatiles. |
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| DC5895 | Apigenin | A plant flavonoid that has been found to inhibit cell proliferation by arresting the cell cycle at the G2/M phase. |
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| DC5880 | Piceatannol | A plant metabolite possessing anti-leukemic activity; inhibits the non-receptor kinases, Syk and Lck. |
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| DC22782 | MDL-72527 Featured | A polyamine oxidase (PAO) inhibitor that inhibits spermine oxidase and N1-acetylpolyamine oxidase with IC50 of 6.1 and 0.02 uM, respectively. |
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| DC22387 | Nystatin | A polyene antifungal antibiotic that works by disrupting the cell membrane of the fungal cells.. |
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| DC22957 | RU-TRAAK-1 | A poorly reversible TRAAK inhibitor, shows no activity for non-K2P channels (Kv1.2, Slo1 and GIRK2).. |
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| DC22647 | NU-7163 | A poten and selective, ATP-competitive DNA-PK inhibitor with IC50 of 0.19 uM, Ki of 24 nM. |
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| DC20911 | Omuralide Featured | A potent 20S proteasome inhibitor with IC50 of 49 nM (inhibition of proteasomal chymotrypsin-like proteolytic activity).. |
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| DC21726 | TAK-802 | A potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM. |
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| DC21727 | TAK-802 hydrochloride | A potent acetylcholinesterase (AChE) inhibitor with IC50 of 1.3 nM. |
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| DC11614 | ENT1-IN-39 | A potent adenosine transport activity of ENT-1 with IC50 of 26.9 nM. |
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| DC20957 | TCDD | A potent AHR (aryl hydrocarbon receptor) agonist that induces degradation of AhR by the ubiquitin-proteasome pathway. |
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| DC23997 | Aleglitazar | A potent and balanced dual PPARα/γ agonist (EC50= 50/21 nM). |
|
| DC22969 | BC-54 | A potent and biologically-active PDE4/7 inhibitor with IC50 of 50-100 nM for PDE4A/B/D, and 140 nM for both PDE7A/B. |
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| DC20804 | BMS-204352 | A potent and effective calcium-sensitive opener of maxi-K potassium channels (maxi-K) with EC50 of 392 nM at -48.4 mV in HEK293 isolated outside-out membrane patches. |
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| DC22960 | ICA-105574 Featured | A potent and efficacious hERG channel activator steeply potentiates current amplitudes more than 10-fold with EC50 of 0.5 uM. |
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| DC20835 | BRD-7880 | A potent and highly specific inhibitor of Aurora B and Aurora C with IC50 of 7 and 12 nM respectively, with less activity against Aurora A (IC50>2 uM). |
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| DC22627 | Trametinib DMSO solvate Featured | A potent and highly specific MEK1/2 inhibitor with IC50 of 0.92 nM/1.8 nM. |
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| DC22496 | W-54011 | A potent and orally active non-peptide C5a receptor (CD88. |
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| DC22772 | ANI-7 | A potent and selective (up to 263-fold) inhibitor of breast cancer cells with GI50 of 0.5 uM (MCF-7), via activation the aryl hydrocarbon receptor (AhR) pathway. |
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| DC22622 | WAY-100635 | A potent and selective 5-HT1A receptor antagonist. |
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| DC21471 | PF-03246799 | A potent and selective 5-HT2C receptor agonist with EC50 of 190 nM, with excellent selectivity for 5-HT2C over 5-HT2A. |
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| DC22368 | Alosetron | A potent and selective 5-HT3 receptor antagonist has been shown to be beneficial in the treatment of irritable bowel syndrome.. |
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| DC23952 | GR-79236 Featured | GR79236 is a highly potent and selective adenosine A1 receptor agonist (Ki = 3.1 nM) that has analgesic and anti-inflammatory actions in humans and animals. |
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| DC20655 | AM-1221 | A potent and selective agonist for the cannabinoid receptor CB1 with Ki of 0.28 nM, 180-fold selectivity over CB2.. |
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| DC22498 | A-443654 Featured | A potent and selective Akt inhibitor with Ki of 0.16 nM for Akt1. |
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| DC23832 | ALK5-IN-16i | A potent and selective ALK5 inhibitor with IC50 of 5.5 nM, displays 300-fold selecitvity over ALK3. |
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| DC22583 | AMD-070 hydrochloride(Mavorixafor) Featured | A potent and selective antagonist of CXCR4 with IC50 of 13 nM in a CXCR4 125I-SDF inhibition binding assay. |
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| DC22376 | Pitolisant oxalate | A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM. |
|
| DC22377 | Pitolisant | A potent and selective antagonist of H3 receptor with Ki/EC50 of 0.16/1.5 nM. |
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