DCC0995 |
Bin-01-07-07 |
Novel USP28 inhibitor |
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DCC0996 |
Bio-0554019 |
Novel selective RORgamma inhibitor, selectively inhibiting Th17 differentiation and RORgamma signature gene expression |
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DCC0997 |
Bipbipu |
Novel heparanase inhibitor |
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DCC0998 |
Biph(2,3',4,5',6)p5 |
Potent inhibitor of SHIP-2 catalytic activity; Novel inositol polyphosphate surrogate modulating Ca responses in rat hepatocytes |
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DCC0999 |
Biphalin |
Potent peptide opioid receptor agonist, alleviating LPS-Induced activation in rat primary microglial cultures in opioid receptor-dependent and receptor-independent manners |
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DCC1000 |
Bis-2-ai Adjuvant-2 |
Novel adjuvant to repurpose azithromycin for use against Pseudomonas aeruginosa, exhibiting a 1024-fold reduction in the minimum inhibitory concentration of azithromycin in vitro and displays activity in a Galleria mellonella model of infection |
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DCC1001 |
Bis-5-methyl-cyclosal-d4tmp |
Novel anti-HIV active dimeric prodrug of 2‘,3‘-dideoxy-2‘,3‘-didehydrothymidine monophosphate (d4TMP) |
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DCC1002 |
Bisaramil |
Class I antiarrhythmic agent with chronotropic, inotropic, dromotropic and coronary vasodilator effects, potently blocking sodium channel |
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DCC1003 |
Bis-cyclosal-d4tmp |
Novel anti-HIV active dimeric prodrug of 2‘,3‘-dideoxy-2‘,3‘-didehydrothymidine monophosphate (d4TMP) |
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DCC1004 |
Bisdionin F |
Selective hAMCase Inhibitor |
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DCC1005 |
Bisindole-pbd |
Novel inhibitor of angiogenesis by regulating STAT3 and VEGF in breast cancer cells |
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DCC1006 |
Bisleuconothine A |
Novel and selective Wnt signaling inhibitor |
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DCC1007 |
bis-n-norgliovictin |
Novel inhibitor of LPS-induced inflammation in macrophages, improving survival in sepsis |
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DCC1008 |
Bisoctrizole |
UV stabilizer |
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DCC1009 |
Bis-salicyl Fumarate |
Potent activator of the Neh2-luc reporter |
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DCC1010 |
Bisthianostat |
Novel Orally Efficacious Pan-HDAC Inhibitor |
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DCC1011 |
Bitc-sg |
Inactivator of GSTP1>GST P1-1 through the covalent modification of two Cys47 residues per dimer and one Cys101 |
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DCC1012 |
Bit-l15 |
Novel potent antagonist of RORγt function, displaying an increased selectivity for RORγt over RORα and PPARγ compared to the purely orthosteric and allosteric non-PEG-linked parent compounds |
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DCC1013 |
Bix-02188me |
Potent and selective dual inhibitor of MEK5 and ERK5 |
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DCC1014 |
Bjff078 |
Potent inhibitor of recombinant human and mouse Transglutaminase enzyme activity, mainly TG2 and the close related enzyme TG1 |
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DCC1015 |
Bjp-06-005-3 |
Novel potent and selective covalent Pin1 inhibitor |
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DCC1016 |
Bki-1708 |
Novel Bumped-Kinase Inhibitor (BKI) for Cryptosporidiosis Therapy |
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DCC1017 |
Bki-1770 |
Novel Bumped-Kinase Inhibitor (BKI) for Cryptosporidiosis Therapy |
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DCC1018 |
Bki-1812 |
Novel potent and selective bumped kinase inhibitor (BKI) CpCDPK1 IC 50 0.0025 µM |
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DCC1019 |
Bki-1814 |
Novel potent and selective bumped kinase inhibitor (BKI) CpCDPK1 IC 50 0.005 µM |
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DCC1020 |
Bkm1644 |
Novel inhibitor of survivin transcription through a signal transducer and activator of transcription 3 (Stat3)-dependent mechanism, inhibiting tissue expression of survivin and inducing apoptosis in C4-2 skeletal tumor |
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DCC1021 |
Bkm1740 |
Novel effective inhibitor of survivin expression at both the mRNA and protein levels in vitro, significantly reducing survivin in bone metastatic C4-2 tumors |
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DCC1022 |
Bkm1972 |
Novel inhibitor of the expression of anti-apoptotic protein survivin and membrane-bound efflux pump ATP binding cassette B 1 (ABCB1, p-glycoprotein), presumably via signal transducer and activator of transcription 3 (Stat3), inhibiting human prostate canc |
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DCC1023 |
Bkm-570 |
Bradykinin antagonist, causing impressive growth inhibition of lung and prostate tumors, displaying superior in vivo inhibitory effects than convential chemotherapeutic drugs |
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DCC1024 |
Blancoxanthone |
Natural anti-coronavirus agent |
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