DCC1145 |
Br-verapamil Hydrochloride |
Novel Ca V channels blocker, binding in the central cavity of the pore on the intracellular side of the selectivity filter, physically blocking the ion-conducting pathway |
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DCC1146 |
Bryostatin 2 |
Protein kinase C (PKC) activator |
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DCC1147 |
Bsc2118 |
Novel proteasome inhibitor, protecting against cerebral ischaemia through HIF1A accumulation and enhanced angioneurogenesis |
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DCC1148 |
bsc4090 |
Fluorescent probe in vitro and in vivo aiming at a tau-based diagnosis of Alzheimer's disease |
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DCC1149 |
bsc4704 |
Fluorescent probe, binding to neurofibrillary tangles with high contrast and selectivity over amyloid |
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DCC1150 |
Bsc4750 |
Fluorescent probe visualizing neurofibrillary tangles in Alzheimer's disease |
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DCC1151 |
Bsh-in-7 |
Novel potent covalent inhibitor of gut bacterial bile salt hydrolases (BSH) |
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DCC1152 |
Bss-730a |
Novel potent inhibitor of both HIV-1 and HIV-2 replication, being also active against the erythrocytic stages of P. falciparum |
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DCC1153 |
Bta9881 |
Novel respiratory syncytial virus (RSV) fusion inhibitor |
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DCC1154 |
btb02467 |
Novel cell-permeable modulator of cellular morphogenesis in yeast and mammalian cells; Inhibitor of SARS-CoV Mpro activity via intensive H-bond network and hydrophobic interactions |
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DCC1155 |
btb03156 |
Novel cell-permeable modulator of cellular morphogenesis in yeast and mammalian cells |
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DCC1156 |
btb03195 |
Novel activator of PC1/3 and inhibitor of PC2 |
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DCC1157 |
Btgh84 Activator I |
Novel activator of BtGH84, the first experimentally discovered small molecule activator of a glycoside hydrolase |
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DCC1158 |
Bti-a-404 |
Novel selective and potent competitive inverse agonist of human GPR43 |
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DCC1159 |
Btk-in-27 |
Novel potent and selective covalent inhibitor of Bruton’s tyrosine kinase (BTK), targeting a noncatalytic cysteine residue (Cys481) for covalent bond formation |
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DCC1160 |
Btk-in-3 |
Novel potent inhibitor of Bruton’s tyrosine kinase (BTK) |
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DCC1161 |
B-tpmf |
The first small-molecule inhibitor with significant selectivity among the KCa2 channel subtypes |
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DCC1162 |
Btt-3035 |
Novel inhibitor of alpha2beta1 integrin, decreasing average platelet adhesion in individuals with the C/T807T genotype but not in those harboring C807C |
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DCC1163 |
Btx-yne |
Novel unique Na V modulator, acting as a conspicuous outlier, eliminating fast but not slow inactivation |
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DCC1164 |
Btz-n3 |
Novel effective reversible and noncovalent inhibitor of DprE1. |
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DCC1165 |
Btzo-4 |
Negative control for BTZO-1 |
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DCC1166 |
Bu99008 |
Ligand of the Imidazoline(2) binding site (I 2 BS), showing very good affinity for the I 2 BS (K i of 1.4 nM; K d = 1.3 nM), good selectivity compared with the α 2 -adrenoceptor (909-fold) |
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DCC1167 |
Bucinnazine |
Potent and selective agonist of μ-opioid receptor (MOR) with relatively low affinity for the δ-opioid receptor and the κ-opioid receptor |
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DCC1168 |
Budralazine |
Direct-acting vasodilator with anti-tachycardiac effect |
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DCC1169 |
Bulgecin A
Featured
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Bulgecin A is an inhibitor of binuclear metallo-beta-lactamases and Lytic transglycosolase. |
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DCC1170 |
Butafenacil |
Potent inducer of anemia |
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DCC1171 |
Butylcycloheptyl Prodiginine |
Natural inhibitor of microRNA-21, reducing growth of cancer cells |
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DCC1172 |
Bvt-116429 |
Novel 11β-HSD1 inhibitor |
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DCC1173 |
bvt-2733 Hydrochloride |
Selective 11beta-hydroxysteroid dehydrogenase type 1 (11betaHSD1) inhibitor |
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DCC1174 |
Bw2258u89 |
Novel BB2 receptor antagonist. attenuating the feeding responses evoked by exogenous gastrin releasing peptide-29 |
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