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CCDC(TGR5-Receptor-Agonist)

  Cat. No.:  DC7319   Featured
Chemical Structure
1197300-24-5
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Field of application
CCDC is a otent, selective TGR5 G-protein coupled receptor agonist (pEC50 = 6.8).
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1197300-24-5
Chemical Name: 4-Isoxazolecarboxamide, 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethyl-
Synonyms: 4-Isoxazolecarboxamide, 3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethyl-;3-(2-Chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethyl-1,2-oxazole-4- carboxamide;3-(2-chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethyl-4-Isoxazolecarboxamide;3-(2-Chlorophenyl)-N-(4-chlorophenyl)-N,5-dimethylisoxazole-4-carboxamide;TGR5;TGR5 Receptor Agonist
SMILES: ClC1=CC=CC=C1C2=NOC(C)=C2C(N(C)C3=CC=C(Cl)C=C3)=O
Formula: C18H14N2O2Cl2
M.Wt: 361.22196
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: TGR5 Receptor Agonist, a potent TGR5(GPCR19) agonist, showed improved potency in the U2-OS cell assay (pEC50 = 6.8) and in melanophore cells (pEC50 = 7.5).
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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