Citarinostat(ACY-241)|cas 1316215-12-9|DC Chemicals

Cas No.:	1316215-12-9
Chemical Name:	Citarinostat
Synonyms:	2-((2-Chlorophenyl)(phenyl)amino)-N-(7-(hydroxyamino)-7-oxoheptyl)pyrimidine-5-carboxamide;ACY-241;Citarinostat;2-?[(2-?chlorophenyl)?phenylamino]?-?N-?[7-?(hydroxyamino)?-?7-?oxoheptyl]?-5-?Pyrimidinecarboxamid?e;ACY241;HDAC-IN-2;2-(N-(2-chlorophenyl)anilino)-N-[7-(hydroxyamino)-7-oxoheptyl]pyrimidine-5-carboxamide;441P620G3P;Citarinostat [USAN];Citarinostat (USAN);AK160199;2-[(2-Chlorophenyl)phenylamino]-N-[7-(hydroxyamino)-7-oxoheptyl]-5-pyrimidinecarboxamide;2-((2-Chlorophenyl)phenylamino)-N-(7-(hydroxyamino)-7-oxoheptyl)-5-pyrimidinecarboxamide;5
SMILES:	ClC1=C([H])C([H])=C([H])C([H])=C1N(C1C([H])=C([H])C([H])=C([H])C=1[H])C1N=C([H])C(=C([H])N=1)C(N([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C([H])([H])C(N([H])O[H])=O)=O
Formula:	C₂₄H₂₆ClN₅O₃
M.Wt:	467.9479
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

Citarinostat is a HDAC6 specific inhibitor, with IC50 of 4 nM and 76 nM for HDAC6 and HDAC3, respectively.IC50 value: 4 nM (HDAC6), 76 nM (HDAC3)Target: HDACThe detailed information please refer to WO2015061684A1 and 2015054197A1.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101
2018-0101

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