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KUNG94

  Cat. No.:  DC11616  
Chemical Structure
2134571-29-0
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More than 5000 active chemicals with high quality for research!
Field of application
A potent, selective Grp94 inhibitor with IC50 of 8 nM.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2134571-29-0
Chemical Name: (5-(4-fluorobenzyl)-2,4-dihydroxyphenyl)(isoindolin-2-yl)methanone
Synonyms: KUNG-94;KUNG 94
SMILES: C(C1=CC(CC2=CC=C(F)C=C2)=C(O)C=C1O)(N1CC2=C(C1)C=CC=C2)=O
Formula: C22H18FNO3
M.Wt: 363.388
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: A potent, selective Grp94 inhibitor with IC50 of 8 nM; displays 10-fold selecticity over Hsp90α; shows antiproliferative activity against RPMI8226 cells with Gi50 of 1.4 uM, reduces LRP6 levels and induces apoptosis.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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