M-COPA |CAS 861718-91-4|DC Chemicals

Cas No.:	861718-91-4
Chemical Name:	(2E,4E)-5-((1S,2S,4aR,6R,7S,8S,8aS)-7-hydroxy-2,6,8-trimethyl-1,2,4a,5,6,7,8,8a-octahydronaphthalen-1-yl)-2-methyl-N-(pyridin-3-yl-methyl)penta-2,4-dienamide
Synonyms:	AMF-26;AMF26;2-Methylcoprophilinamide
SMILES:	O=C(NCC1=CC=CN=C1)/C(C)=C/C=C/[C@H]2[C@@H](C)C=C[C@@]3([H])C[C@@H](C)[C@H](O)[C@@H](C)[C@]23[H]
Formula:	C₂₅H₃₄N₂O₂
M.Wt:	394.559
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

A small-molecule compound that disrupts the Golgi apparatus by inhibiting the activation of ADP-ribosylation factor 1 (ARF1); inhibits transport of Stx from the plasma membrane to the Golgi apparatus and suppresses degradation of anti-apoptotic proteins and the activation of caspases, inhibits Stx-induced apoptosis in E, coli; inhibits cell surface expression of MET protein and exhibits antitumor activity against MET-addicted gastric cancers.

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

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(2E,4E)-5-((1S,2S,4aR,6R,7S,8S,8aS)-7-hydroxy-2,6,8-trimethyl-1,2,4a,5,6,7,8,8a-octahydronaphthalen-1-yl)-2-methyl-N-(pyridin-3-yl-methyl)penta-2,4-dienamide