CJ-13610|cas 179420-17-8|DC Chemicals

Cas No.:	179420-17-8
Chemical Name:	2H-Pyran-4-carboxamide,tetrahydro-4-[3-[[4-(2-methyl-1H-imidazol-1-yl)phenyl]thio]phenyl]-
Synonyms:	2H-Pyran-4-carboxamide,tetrahydro-4-[3-[[4-(2-methyl-1H-imidazol-1-yl)phenyl]thio]phenyl]-;4-[3-[4-(2-methylimidazol-1-yl)phenyl]sulfanylphenyl]oxane-4-carboxamide
SMILES:	CC1=NC=CN1C1C=CC(SC2=CC=CC(C3(C(N)=O)CCOCC3)=C2)=CC=1
Formula:	C₂₂H₂₃N₃O₂S
M.Wt:	393.501923799515
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

CJ-13610 is a potent 5-Lipoxygenase (5-LO) inhibitor that suppresses 5-LO product formation with IC50 of 70 nM; demonstrates antihyperalgesic activity in inflammatory pain models including the acute carrageenan model and the chronic inflammatory model.AsthmaPhase 2 Discontinued

MSDS

COA

LOT NO.	DOWNLOAD
2018-0101

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