SU 16f|cas 251356-45-3|DC Chemicals

Cas No.:	251356-45-3
Chemical Name:	3-[2,4-dimethyl-5-[(2-oxo-6-phenyl-1H-indol-3-ylidene)methyl]-1H-pyrrol-3-yl]propanoic acid
Synonyms:	1H-Pyrrole-3-propanoic acid, 5-[(1,2-dihydro-2-oxo-6-phenyl-3H-indol-3-ylidene)methyl]-2,4-dimethyl-;3-[2,4-dimethyl-5-[(2-oxo-6-phenyl-1H-indol-3-ylidene)methyl]-1H-pyrrol-3-yl]propanoic acid;SU 16F;3-[2,4-Dimethyl-5-(2-oxo-6-phenyl-1,2-dihydroindol-3-ylidenemethyl)-1H-pyrrol-3-yl]-propionic acid;3-{2,4-Dimethyl-5-[(2-oxo-6-phenyl-1,2-dihydro-3H-indol-3-ylidene)methyl]-1H-pyrrol-3-yl}propanoic acid;SU16f
SMILES:	C1=C2/C(=C/C3NC(C)=C(CCC(=O)O)C=3C)/C(=O)NC2=CC(C2C=CC=CC=2)=C1
Formula:	C₂₄H₂₂N₂O₃
M.Wt:	386.443086147308
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

SU 16f is a potent and selective PDGFRβ inhibitor with IC50 of 10 nM, displays >14-fold, >229-fold and >10,000-fold selectivity over VEGFR2, FGFR1 and EGFR respectively; inhibits proliferation of HUVEC and NIH3T3 cells in vitro (IC50 =0.11 uM).

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101
2018-0101

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