RO 27-3225

  Cat. No.:  DC22215   Featured
Chemical Structure
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More than 5000 active chemicals with high quality for research!
Field of application
RO 27-3225 (RO27-3225, RO 273225) is a potent, selective melanocortin melanocortin receptor MC4R agonist with EC50 of 1 nM, >30-fold selectivity over MC3R.
Cas No.:
Chemical Name: Butir-His-D-Phe-Arg-Trp-Sar-NH2 trifluoracetate salt
Synonyms: RO 27-3225|RO27-3225;RO 273225
SMILES: CCCC(=O)N[C@@H](CC1=CN=CN1)C(=O)N[C@@H](CC2=CC=CC=C2)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC3=CNC4=CC=CC=C43)C(=O)N(C)CC(=O)N
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: RO 27-3225 (RO27-3225, RO 273225) is a potent, selective melanocortin melanocortin receptor MC4R agonist with EC50 of 1 nM, >30-fold selectivity over MC3R; shows some activity at the MC1 receptor (EC50=8 nM), reverses hemorrhagic shock, reduces multiple organ damage, and improves survival.ObesityDiscontinued
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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