RO 27-3225|RO27-3225| MC4R agonist|DC Chemicals

Cas No.:
Chemical Name:	Butir-His-D-Phe-Arg-Trp-Sar-NH2 trifluoracetate salt
Synonyms:	RO 27-3225\|RO27-3225;RO 273225
SMILES:	CCCC(=O)N[C@@H](CC1=CN=CN1)C(=O)N[C@@H](CC2=CC=CC=C2)C(=O)N[C@@H](CCCN=C(N)N)C(=O)N[C@@H](CC3=CNC4=CC=CC=C43)C(=O)N(C)CC(=O)N
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

RO 27-3225 (RO27-3225, RO 273225) is a potent, selective melanocortin melanocortin receptor MC4R agonist with EC50 of 1 nM, >30-fold selectivity over MC3R; shows some activity at the MC1 receptor (EC50=8 nM), reverses hemorrhagic shock, reduces multiple organ damage, and improves survival.ObesityDiscontinued

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

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