Bromocriptine mesylate| CAS 22260-51-1

Cas No.:	22260-51-1
Chemical Name:	Bromocriptine mesylate
Synonyms:	Bromocriptine mesylate;2-Bromo-alpha-ergocryptine methanesulfonate;(+)-2-Bromo-12'-hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)ergotaman-3',6'-18-trione methanesulfonate salt;2-Bromo α-Ergocryptine Mesylate;2-BroMo-α-ergocryptine Methanesulfonate salt;Bromocriptine (mesylate);Bromocriptine Methanesulphonate;CB-154;Bromocriptine mesilate;Parlodel;(+)-2-Bromo-12′-hydroxy-2′-(1-methylethyl)-5′-(2-methylpropyl)ergotaman-3′,6′-18-trione methanesulfonate salt;(+)-Bromocriptine methanesulfonate salt;Bromocriptine mesylate salt;CAS-22260-51-1;BROMOCRIPTINE MESILATE (MART.);CB 154 methanesulfonate (salt);2-Bromoergocryptine monomethanesulfonate (salt);BROMOCRIPTINE MESYLATE;Bromocriptine mesylate (USP);2-Bromo alpha-Ergocryptine Mesylate;Tox21_500171;SR-01000597796-1;DTXSID6020197;.alpha.-Ergocryptine, methanesulfonate;NCGC00260856-01;B 2134;2-Bromine-alpha-ergocryptine methanesulfonate;(5'alpha)-2-bromo-12'-hydroxy-5'-(2-methylpropyl)-3',6',18-trioxo-2'-(propan-2-yl)ergotaman methanesulfonate (salt);C32H40BrN5O5.CH3SO3H;D81822;Bromocriptine mesylate [USAN];2-Bromo-alpha-ergocryptine mesylate;BROMOCRIPTINEMESYLATE;BROMOCRIPTINE MESYLATE [USP-RS];BROMOCRIPTINE MESILATE (EP MONOGRAPH);ERGOTAMAN-3',6',18-TRIONE, 2-BROMO-12'-HYDROXY-2'-(1-METHYLETHYL)-5'-(2-METHYLPROPYL)-, MONOMETHANESULFONATE (SALT), (5'.ALPHA.)-;2-Bromoergocryptine Mesylate;2-Bromo-alpha-ergokryptine-mesilate;CCG-220121;Prestwick_771;22260-51-1;Ergotaman-3',6',18-trione, 2-bromo-12'-hydroxy-2'-(1-methylethyl)-5'-(2-methylpropyl)-, monomethanesulfonate (salt), (5'alpha)-;BROMOCRIPTINE MESYLATE [VANDF];BROMOCRIPTINE MESYLATE [USP MONOGRAPH];2-Bromo ?-Ergocryptine Mesylate;Cycloset;2-BROMOERGOCRYPTINE MONOMETHANESULPHONATE (SALT);HMS3712I04;Tox21_303597;CS-6048;Bromocriptine mesylate (USAN:USP);(+)-Bromocriptine methanesulfonate;SR-01000075356;AKOS015896276;2-Bromo-12'-hydroxy-5'alpha-isobutyl-2'-isopropylergotaman-3',6',18-trione monomethanesulphonate;BROMOCRIPTINE MESYLATE (USP MONOGRAPH);EU-0100171;Pravidel;NSC169774;BROMOCRIPTINE MESILATE [EP MONOGRAPH];NSC-755915;SR-01000597796;DTXCID00197;Bromocryptine methanesulfonate;ERGOTAMAN-3',6',18-TRIONE, 2-BROMO-12'-HYDROXY-2'-(1-METHYLETHYL)-5'-(2-METHYLPROPYL)-, MONOMETHANESULPHONATE (SALT), (5'alpha)-;BROMOCRIPTINE MESILATE [MART.];2-Bromo-alpha-ergokryptine-mesilate [German];BB164266;Q27105974;Bromocriptine mesilate (JP17);BROMOCRIPTINE MESILATE [WHO-DD];LP00171;BROMOCRIPTINE MESYLATE [ORANGE BOOK];Bromocriptine mesylate [USAN:USP];HMS3411K09;2-Bromo-.alpha.-ergocryptine monomethanesulfonate;EINECS 244-881-1;HB1813;HMS1568I04;Parlodel (TN);CHEMBL1200503;CCG-221475;NCGC00257268-01;Bromocryptine mesylate;Bagren;2-Bromo-a-ergocryptine methanesulfonate salt;Bromocriptine methanesulfonate;BROMOCRIPTINE MESILATE [JAN];SR-01000075356-1;Bromocriptine mesylate- Bio-X;Bromergon;alpha-Ergocryptine, 2-bromo-, methanesulfonate;NSC 7559...
SMILES:	[H][C@@]12CC3=C(Br)NC4=CC=CC(C1=C[C@@H](C(N[C@@]5(C(C)C)C(N6[C@@H](CC(C)C)C(N7CCC[C@]7([C@]6(O)O5)[H])=O)=O)=O)CN2C)=C43.OS(=O)(C)=O
Formula:	C₃₂H₄₀N₅O₅Br^.CH₄O₃S
M.Wt:	750.700160000001
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

Bromocriptine (CB-154) is a dopamine D2 receptor agonist (Ki=3 nM) and and various serotonin receptors, also inhibits the release of glutamate by reversing the glutamate GLT1 transporter; decreases body fat in animal and human models and increases lean muscle mass, improves glucose intolerance and insulin resistance, and reduces triglycerides and free fatty acids; also induces apoptosis and decreases colony formation in AML cells, shows synergy with standard agents and selectivity for the leukemic cell; reduces hyperphagia and adiposity in rats with diet-induced obesity.DiabetesApproved

MSDS

COA

LOT NO.	DOWNLOAD

2018-0101

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