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GSK-805

  Cat. No.:  DC33598   Featured
Chemical Structure
1426802-50-7
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More than 5000 active chemicals with high quality for research!
Field of application
GSK805, also known as ROR gamma-t-IN-1, is a potent, orally bioavailable retinoid-related orphan receptor gamma t (RORγt) inverse agonist that interacts with the receptor's putative ligand binding domain without exerting significant effects on DNA binding.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1426802-50-7
Chemical Name: N-[2,6-dichloro-2'-(trifluoromethoxy)[1,1'-biphenyl]-4-yl]-4-(ethylsulfonyl)-benzeneacetamide
Synonyms: GSK805; GSK 805; GSK-805; ROR gamma-t-IN-1; RORγt Inverse Agonist II;
SMILES: O=C(NC1=CC(Cl)=C(C2=CC=CC=C2OC(F)(F)F)C(Cl)=C1)CC3=CC=C(S(=O)(CC)=O)C=C3
Formula: C23H18Cl2F3NO4S
M.Wt: 532.3552
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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