JTC-801|cas 244218-51-7|DC Chemicals|Price|Buy

Cas No.:	244218-51-7
Chemical Name:	N-(4-amino-2-methylquinolin-6-yl)-2-((4-ethylphenoxy)methyl)benzamide hydrochloride
Synonyms:	JTC 801; JTC801
SMILES:	NC1=CC(C)=NC2=C1C=C(NC(C3=C(COC4=CC=C(C=C4)CC)C=CC=C3)=O)C=C2.[H]Cl
Formula:	C₂₆H₂₅N₃O₂^.HCl
M.Wt:	447.96
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO

Description:

JTC-801 displays about 12.5-, 129-, and 1055-fold selectivity For ORL1 receptor (Ki = 8.2 nM) over μ-, κ-, and δ-opioid receptors, respectively. JTC-801 does not inhibit Forskolin-stimulated cyclic AMP accumulation in human ORL1 receptor-expressing HeLa

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2018-0101

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