PSMA-617 Linker|CAS 1703768-74-4|DC Chemicals

Cas No.:	1703768-74-4
Chemical Name:	Vipivotide tetraxetan Ligand-Linker Conjugate
Synonyms:	PSMA-617 Linker;Vipivotide tetraxetan Linker;JUN68744;(((S)-5-((S)-2-((1r,4S)-4-(aminomethyl)cyclohexane-1-carboxamido)-3-(naphthalen-2-yl)propanamido)-1-carboxypentyl)carbamoyl)-L-glutamic acid;Vipivotide tetraxetan Ligand-Linker Conjugate
SMILES:	O=C(C1CCC(CN)CC1)N[C@H](C(NCCCC[C@@H](C(=O)O)NC(N[C@H](C(=O)O)CCC(=O)O)=O)=O)CC1C=CC2C=CC=CC=2C=1
Formula:	C₃₃H₄₅N₅O₉
M.Wt:	655.738508939743
Purity:	>98%
Sotrage:	-20
Publication:	[1]. Benešová M, et al. Albumin-Binding PSMA Ligands: Optimization of the Tissue Distribution Profile. Mol Pharm. 2018 Mar 5;15(3):934-946.

Description:

Vipivotide tetraxetan Ligand-Linker Conjugate (PSMA-617 Ligand-Linker Conjugate) is composed of a linker and Glutamate-urea-Lysine, can be used to synthesize Vipivotide tetraxetan (PSMA-617). Glutamate-urea-Lysine is is the selective pharmacophore to bind to prostate specific membrane antigen (PSMA).

MSDS

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MSDS_15922_DC33611_1703768-74-4

COA

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