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LIT-001 trifluoroacetate

  Cat. No.:  DC12434   Featured
Chemical Structure
2245072-21-1
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More than 5000 active chemicals with high quality for research!
Field of application
LIT-001 trifluoroacetate (LIT001) is the first nonpeptide Oxytocin receptor (OT-R) agonist with EC50 of 55 nM, Emax=96%.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2245072-21-1
Chemical Name: (S)-2-(Dimethylcarbamothioyl)-N-(2-methyl-4-(1-methyl-1,4,5,10-tetrahydrobenzo[b]pyrazolo[3,4-e][1,4]diazepine-5-carbonyl)benzyl)pyrrolidine-1-carboxamide 2,2,2-trifluoroacetate
Synonyms: (2S)-2-(Dimethylcarbamothioyl)-N-[[2-methyl-4-(1-methyl-4,10-dihydropyrazolo[4,3-c][1,5]benzodiazepi;LIT-001;D81367;(S)-2-(Dimethylcarbamothioyl)-N-(2-methyl-4-(1-methyl-1,4,5,10-tetrahydrobenzo[b]pyrazolo[3,4-e][1,4;(2S)-2-(dimethylcarbamothioyl)-N-[[2-methyl-4-(1-methyl-4,10-dihydropyrazolo[4,3-c][1,5]benzodiazepine-5-carbonyl)phenyl]methyl]pyrrolidine-1-carboxamide;2,2,2-trifluoroacetic acid;LIT-001 trifluoroacetate;LIT-001 TFA;HY-124733A;MFCD32644853;2245072-21-1;BS-16090;(2S)-2-(dimethylcarbamothioyl)-N-[(2-methyl-4-{4-methyl-2,4,5,9-tetraazatricyclo[8.4.0.0(3),?]tetradeca-1(14),3(7),5,10,12-pentaene-9-carbonyl}phenyl)methyl]pyrrolidine-1-carboxamide; trifluoroacetic acid;CS-0087519;AKOS037648947;(S)-2-(Dimethylcarbamothioyl)-N-(2-methyl-4-(1-methyl-1,4,5,10-tetrahydrobenzo[b]pyrazolo[3,4-e][1,4]diazepine-5-carbonyl)benzyl)pyrrolidine-1-carboxamide 2,2,2-trifluoroacetate;C30H34F3N7O4S;EX-A4570
SMILES: S=C([C@@H]1CCCN1C(NCC1C=CC(=CC=1C)C(N1C2C=CC=CC=2NC2=C(C=NN2C)C1)=O)=O)N(C)C.FC(C(=O)O)(F)F
Formula: C30H34F3N7O4S
M.Wt: 645.695675373077
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: LIT-001 trifluoroacetate (LIT001) is the first nonpeptide Oxytocin receptor (OT-R) agonist with EC50 of 55 nM, Emax=96%; efficiently relieved social interaction deficits in Oprm1−/− mice, a mouse model of autism.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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