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LIT-001 trifluoroacetate

  Cat. No.:  DC12434  
Chemical Structure
2245072-21-1
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More than 5000 active chemicals with high quality for research!
Field of application
LIT-001 trifluoroacetate (LIT001) is the first nonpeptide Oxytocin receptor (OT-R) agonist with EC50 of 55 nM, Emax=96%.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2245072-21-1
Chemical Name: (S)-2-(Dimethylcarbamothioyl)-N-(2-methyl-4-(1-methyl1,4,5,10-tetrahydrobenzo[b]pyrazolo[3,4-e][1,4]diazepine-5- carbonyl)benzyl)pyrrolidine-1-carboxamide, trifluoroacetate
Synonyms: LIT001
SMILES: N(C(NCC1=CC=C(C(N2CC3C=NN(C)C=3NC3=CC=CC=C23)=O)C=C1C)=O)1CCC[C@@H]1C(=S)N(C)C.C(O)(=O)C(F)(F)F
Formula: C30H34F3N7O4S
M.Wt: 645.702
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: LIT-001 trifluoroacetate (LIT001) is the first nonpeptide Oxytocin receptor (OT-R) agonist with EC50 of 55 nM, Emax=96%; efficiently relieved social interaction deficits in Oprm1−/− mice, a mouse model of autism.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
Cat. No. Product name Field of application
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