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Perospirone

  Cat. No.:  DC29051   Featured
Chemical Structure
150915-41-6
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Field of application
Perospirone (SM-9018 free base) is an orally active antagonist of 5-HT2A receptor (Ki=0.6 nM) and dopamine D2 receptor (Ki=1.4 nM), and also a partial agonist of 5-HT1A receptor (Ki=2.9 nM). Perospirone is an atypical antipsychotic drug and has the potential for schizophrenic disease treatment.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 150915-41-6
Chemical Name: Perospirone
Synonyms: 1H-Isoindole-1,3(2H)-dione,2-[4-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]butyl]hexahydro-,(3aR,7aS)-rel-;1H-Isoindole-1,3(2H)-dione,2-[4-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]butyl]hexahydro-,(3...;PEROSPIRINE;[14C]-Perospirone;[3H]-Perospirone;AC1L3H05;CHEMBL1472975;cis-2-[4-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]butyl]-hexahydro-1H-isoindole-1,3(2H)-dione;Lullan;M813;Perospirone;SureCN120579;UNII-N303OK87DT;PEROSPIRONE HCL;cis-N-[4-[4-(1,2-Benzisothiazol-3-yl)-1-piperazinyl]butyl]-1,2-cyclohexanedicarboximide;(1R,2S)-N-[4-[4-(1,2-Benzisothiazole-3-yl)-1-piperazinyl]butyl]cyclohexane-1,2-dicarbimide;1H-Isoindole-1,3(2H)-dione, 2-[4-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]butyl]hexahydro-, cis-;(3aα,7aα)-2-[4-[4-(1,2-Benzisothiazol-3-yl)-1-piperazinyl]butyl]hexahydro-1H-isoindole-1,3(2H)-dione;(3aS,7aR)-2-[4-[4-(1,2-Benzothiazol-3-Yl)Piperazin-1-Yl]Butyl]-3a,4,5,6,7,7a-Hexahydroisoindole-1,3-Dione;1H-Isoindole-1,3(2H)-dione, 2-[4-[4-(1,2-benzisothiazol-3-yl)-1-piperazinyl]butyl]hexahydro-, (3aR,7aS)-rel- (9CI);A809087;(3aR,7aS)-2-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione;Perospirone;SM-9018 (free base);HMS3715H10;HY-B0731A;GTPL7556;s5185;MRF-0000147;DB08922;Lullan (Japan);CHEBI:94777;AS-14845;NS00071002;DTXSID2048163;(3aR,7aS)-2-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione;CS-0019906;SCHEMBL120579;PEROSPIRONE [WHO-DD];cis-N-(4-(4-(1,2-Benzisothiazol-3-yl)-1-piperazinyl)butyl)-1,2-cyclohexanedicarboximide;N303OK87DT;NCGC00164567-01;CCG-221234;(3aR,7aS)-2-(4-(4-(benzo[d]isothiazol-3-yl)piperazin-1-yl)butyl)hexahydro-1H-isoindole-1,3(2H)-dione;Q6590349;(3aR,7aS)-2-[4-[4-(1,2-benzothiazol-3-yl)-1-piperazinyl]butyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione;cis-N-[4-[4-(1,2-benzisothiazole-3-yl)-1-piperazinyl]butyl]cyclohexane-1,2-dicarboximide;AKOS025311209;PEROSPIRONE [MI];1H-Isoindole-1,3(2H)-dione, 2-(4-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)butyl)hexahydro-, (3aR,7aS)-rel-;AB00698486-07;Perospirone [INN];1H-Isoindole-1,3(2H)-dione, 2-(4-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)butyl)hexahydro-, cis-;J-008757;150915-41-6;SM-9018 free base;perospirona;DB-289872;Perospirone Free Base;(3aR,7aS)-2-{4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl}-octahydro-1H-isoindole-1,3-dione;2-(4-(4-(1,2-benzisothiazol-3-yl)-1-piperazinyl)butyl)hexahydro-1H-isoindole-1,3-(2H)-dione;DTXCID3028138;GLXC-21078;(3aS,7aR)-2-(4-(4-(1,2-benzothiazol-3-yl)piperazin-1-yl)butyl)-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione;BRD-K85503079-001-02-8;perospironum;(3aR,7aS)-2-(4-(4-(1,2-benzothiazol-3-yl)piperazin-1-yl)butyl)-octahydro-1H-isoindole-1,3-dione;(3aS,7aR)-2-[4-[4-(1,2-benzothiazol-3-yl)piperazin-1-yl]butyl]-3a,4,5,6,7,7a-hexahydroisoindole-1,3-dione;G12739;BRD-K85503079-001-01-0;Perospirine;PEROSPIRONE
SMILES: C(CCN1C(=O)[C@H]2CCCC[C@H]2C1=O)CN1CCN(C2=NSC3=CC=CC=C23)CC1
Formula: C23H30N4O2S
M.Wt: 426.5749
Purity: 98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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