T5910047 |CAS 950003-29-9|DC Chemicals

Cas No.:	950003-29-9
Chemical Name:	N-{5-(diethylsulfamoyl)thiophen-2-ylmethyl}-4-phenylpiperazine-1-carboxamide
Synonyms:	T5996207;N-((5-(N,N-Diethylsulfamoyl)thiophen-2-yl)methyl)-4-phenylpiperazine-1-carboxamide;T5910047;Z231068704;N-{[5-(diethylsulfamoyl)thiophen-2-yl]methyl}-4-phenylpiperazine-1-carboxamide;N-{5-(diethylsulfamoyl)thiophen-2-ylmethyl}-4-phenylpiperazine-1-carboxamide
SMILES:	S(C1=CC=C(CNC(N2CCN(C3C=CC=CC=3)CC2)=O)S1)(N(CC)CC)(=O)=O
Formula:	C₂₀H₂₈N₄O₃S₂
M.Wt:	436.59132194519
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

T5910047 (T-5910047) is a small molecule inhibitor of MyD88-dependent signaling pathways, disrupts MyD88 homodimeric formation; inhibits SEB-induced inhibition of cytokine production in PBMCs with IC50 of 2-10 uM, also inhibits SEA-induced pro-inflammatory cytokine production, shows no toxicity in primary cells up to 100 uM.

MSDS

COA

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2018-0101

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